The role of 5-HT(1B/1D) receptors in the modulation of 5-hydroxytryptamine levels in the frontal cortex of the conscious guinea pig.

No abstract is available for this paper.

• Publication year

  1997

• Venue

  European Journal of Pharmacology

• Publication date

  1997-05-12

• Fields of study

  Biology, Medicine, Chemistry

• Identifiers
  DOI 10.1016/S0014-2999(97)00156-8PMID 9178651
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites

  2004cited by this paper
• Alignment of receptor nomenclature with the human genome: classification of 5-HT1B and 5-HT1D receptor subtypes.

  1996cited by this paper
• Functional characterization of the 5‐HT terminal autoreceptor in the guinea‐pig brain cortex

  1996cited by this paper
• Evidence that 5‐hydroxytryptamine release in rat dorsal raphé nucleus is controlled by 5‐HT1A, 5‐HT1B and 5‐HT1D autoreceptors

  1995cited by this paper
• The effects of GR127935, a putative 5-HT1D receptor antagonist, on brain 5-HT metabolism, extracellular 5-HT concentration and behaviour in the guinea pig.

  1995cited by this paper
• Effects of the 5-HT1D receptor antagonist GR127935 on extracellular levels of 5-HT in the guinea-pig frontal cortex as measured by microdialysis.

  1995cited by this paper
• 5-HT 1D receptors mediate SKF 99101H-induced hypothermia in the guinea pig

  1995cited by this paper
• An anaesthetic mask for use on guineapigs (Cavia porcellus) in a stereotaxic frame: technical note

  1995cited by this paper
• 5-HT1D as well as 5-HT1A autoreceptors modulate 5-HT release in the guinea-pig dorsal raphé nucleus.

  1994cited by this paper
• Chronic treatment with citalopram facilitates the effect of a challenge dose on cortical serotonin output: role of presynaptic 5-HT1A receptors.

  1994cited by this paper
• Lack of 5-HT1A autoreceptor desensitization following chronic citalopram treatment, as determined by in vivo microdialysis.

  1994cited by this paper
• The use of nitrates, calcium channel blockers and ACE inhibitors in primary care in the Northern Region: a pharmacoepidemiological study.

  1994cited by this paper
• Pindolol induces a rapid improvement of depressed patients treated with serotonin reuptake inhibitors.

  1994cited by this paper
• Effect of acute and repeated administration of 5-HT1A receptor agonists on 5-HT release in rat brain in vivo

  1993cited by this paper
• Terminal Autoreceptor Control of 5‐Hydroxytryptamine Release as Measured by In Vivo Microdialysis in the Conscious Guinea‐Pig

  1992cited by this paper
• Effects of methiothepin on changes in brain serotonin release induced by repeated administration of high doses of anorectic serotoninergic drugs.

  1992cited by this paper
• Pharmacological characteristics of 5‐hydroxytryptamine autoreceptors in rat brain slices incorporating the dorsal raphe or the suprachiasmatic nucleus

  1992cited by this paper
• Desensitization of 5-HT1A autoreceptors by chronic administration of 8-OH-DPAT.

  1992cited by this paper
• Rapid serotonin depletion as a provocative challenge test for patients with major depression: relevance to antidepressant action and the neurobiology of depression.

  1991cited by this paper
• Species differences in presynaptic serotonin autoreceptors: mainly 5-HT1B but possibly in addition 5-HT1D in the rat, 5-HT1D in the rabbit and guinea-pig brain cortex

  1991cited by this paper
• In vivo evidence that 5-hydroxytryptamine (5-HT) neuronal firing and release are not necessarily correlated with 5-HT metabolism.

  1990cited by this paper
• In vivo effects of sumatriptan (GR 43175) on extracellular levels of 5-HT in the guinea pig.

  1990cited by this paper
• Differential responsiveness of the rat dorsal and median raphe 5‐HT systems to 5‐HT1 receptor agonists and p‐chloroamphetamine

  1990cited by this paper
• Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain.

  1989cited by this paper
• A pharmacological analysis of the 5-HT receptor mediating inhibition of 5-HT release in the guinea-pig frontal cortex.

  1988cited by this paper
• Modifications of the Serotonin System by Antidepressant Treatments: Implications for the Therapeutic Response in Major Depression

  1987cited by this paper
• Electrophysiologically-identified serotonin receptors in the rat CNS. Effect of antidepressant treatment.

  1984cited by this paper
• The brain of the guinea pig in stereotaxic coordinates.

  1977cited by this paper
• Use of synthesis inhibitors in defining a role for biogenic amines during imipramine treatment in depressed patients.

  1975cited by this paper
• The treatment of depressive states with G 22355 (imipramine hydrochloride).

  1958cited by this paper
• A preliminary report on marsilid.

  1957cited by this paper
• Mental depression in hypertensive patients treated for long periods with large doses of reserpine.

  1954cited by this paper
• [The action of isonicotinyl-hydrazide used in the treatment of depressive states].

  1952cited by this paper

• Clozapine impaired glucose-stimulated insulin secretion partly by increasing plasma 5-HT levels due to the inhibition of OCT1-mediated hepatic 5-HT uptake in mice

  2024cites this paper
• Altered Serotonin 1B Receptor Binding After Escitalopram for Depression Is Correlated With Treatment Effect

  2024cites this paper
• Multiple facets of serotonergic modulation.

  2021cites this paper
• Effects Of The Antidepressant Drug Vortioxetine On Ventral Pallidal Neuronal Activity, Respiration, And Heart Rate In The Rat

  2021cites this paper
• Serotonergic Regulation of Prefrontal Cortical Circuitries Involved in Cognitive Processing: A Review of Individual 5-HT Receptor Mechanisms and Concerted Effects of 5-HT Receptors Exemplified by the Multimodal Antidepressant Vortioxetine.

  2015cites this paper
• 5-HT Receptor Antagonism Attenuates the Ischemia-Reperfusion Injury After Rabbit Lung Preservation.

  2015cites this paper
• Modifications of plasma 5-HT concentrations during the allergic bronchoconstriction in guinea pigs

  2013cites this paper
• Re view Article NEW INSIGHTS INTO MOLECULAR TARGETS FOR DEPRESSION

  2011cites this paper
• GSK 163090 ) , a Potent , Selective , and Orally Active 5-HT 1 A / B / D Receptor Antagonist

  2010cites this paper
• 5-HT(1B) receptor regulation of serotonin (5-HT) release by endogenous 5-HT in the substantia nigra.

  2010cites this paper
• Discovery of 1-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-2-imidazolidinone (GSK163090), a Potent, selective, and orally active 5-HT1A/B/D receptor antagonist.

  2010cites this paper
• Role of 5‐HT2A, 5‐HT4 and 5‐HT7 receptors in the antigen‐induced airway hyperresponsiveness in guinea‐pigs

  2010cites this paper
• 5-HT1 receptor augmentation strategies as enhanced efficacy: therapeutics for psychiatric disorders.

  2008cites this paper
• Identification and role of serotonin 5-HT1A and 5-HT1B receptors in primary cultures of rat embryonic rostral raphe nucleus neurons.

  2008cites this paper
• Novel 5-HT(1A/1B/1D) receptors antagonists with potent 5-HT reuptake inhibitory activity.

  2008cites this paper
• In vivo/ex vivo and behavioural study on central effects of 5-HT1B/1D and 5-HT1A antagonists in guinea pigs.

  2008cites this paper
• Spatial-specific action of serotonin within the leech midbody ganglion

  2008cites this paper
• Enhanced selective serotonin re-uptake inhibitors as antidepressants: 2004 – 2006

  2007cites this paper
• LES RECEPTEURS 5-HT1B : IMPLICATION DANS LE MECANISME D'ACTION DES ANTIDEPRESSEURS

  2006cites this paper
• SB-616234-A (1-[6-(cis-3,5-dimethylpiperazin-1-yl)-2,3-dihydro-5-methoxyindol-1-yl]-1-[2'methyl-4'-(5-methyl-1,2,3-oxadiazol-3-yl)biphenyl-4-yl]methanone hydrochloride): a novel, potent and selective 5-HT1B receptor antagonist.

  2006cites this paper
• SB-236057-A: a selective 5-HT1B receptor inverse agonist.

  2006cites this paper
• UNIVERSIDADE FEDERAL DO RIO GRANDE DO SUL INSTITUTO DE CIÊNCIAS BÁSICAS DA SÁUDE PROGRAMA DE PÓS-GRADUAÇÃO EM NEUROCIÊNCIAS

  2006cites this paper
• 5-HT1B receptors, ventral orbitofrontal cortex, and aggressive behavior in mice

  2006cites this paper
• Characterisation of the selective 5-HT1B receptor antagonist SB-616234-A (1-[6-(cis-3,5-dimethylpiperazin-1-yl)-2,3-dihydro-5-methoxyindol-1-yl]-1-[2'-methyl-4'-(5-methyl-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methanone hydrochloride): in vivo neurochemical and behavioural evidence of anxiolytic/antidep

  2006cites this paper
• Synthesis and SAR of highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drugs.

  2005cites this paper
• Escalated aggressive behavior: dopamine, serotonin and GABA.

  2005cites this paper
• Innovative approaches for the development of antidepressant drugs: Current and future strategies

  2005cites this paper
• Differential autoreceptor control of extracellular 5-HT in guinea pig and rat: species and regional differences

  2004influential citation
• The effects of selective serotonin reuptake inhibitors on extracellular 5-HT levels in the hippocampus of 5-HT(1B) receptor knockout mice.

  2002cites this paper
• 5-HT1B receptors and serotonin function : microdialysis studies in rats and knockout mice

  2002cites this paper
• Evidence for involvement of protein kinases in the regulation of serotonin synthesis and turnover in the mouse brain in vivo

  2002cites this paper
• Ligands for the investigation of 5-HT autoreceptor function.

  2001cites this paper
• The role of 5‐HT1B receptors in the regulation of serotonin cell firing and release in the rat brain

  2001cites this paper
• Zolmitriptan – a 5-HT1B/D agonist, alcohol, and aggression in mice

  2001cites this paper
• Oral drug self-administration in the home cage of mice: alcohol-heightened aggression and inhibition by the 5-HT1B agonist anpirtoline

  2001cites this paper
• LY393558, a 5-hydroxytryptamine reuptake inhibitor and 5-HT(1B/1D) receptor antagonist: effects on extracellular levels of 5-hydroxytryptamine in the guinea pig and rat.

  2001cites this paper
• Serotonergic effects and extracellular brain levels of eletriptan, zolmitriptan and sumatriptan in rat brain.

  2001cites this paper
• Mechanisms underlying the speed of onset of antidepressant response

  2001cites this paper
• The possible role of 5-HT(1B/D) receptors in psychiatric disorders and their potential as a target for therapy.

  2000cites this paper
• The effect of SB-236057-A, a selective 5-HT1B receptor inverse agonist, on in vivo extracellular 5-HT levels in the freely-moving guinea-pig

  2000cites this paper
• Serotonergic modulation of ethanol-induced electrophysiological depression in young and aged rats.

  2000cites this paper
• Regulation of extracellular concentrations of 5-hydroxytryptamine (5-HT) in mouse striatum by 5-HT(1A) and 5-HT(1B) receptors.

  2000cites this paper
• 5-HT reuptake inhibitors with 5-HT(1B/1D) antagonistic activity: a new approach toward efficient antidepressants.

  2000cites this paper
• Chapter 23 Antidepressant and anxiolytic drugs

  2000cites this paper
• Control of dorsal raphé 5-HT function by multiple 5-HT(1) autoreceptors: parallel purposes or pointless plurality?

  2000cites this paper
• 5-HT1B/D receptors in anxiety

  2000cites this paper
• Amplification of cortical serotonin release: a further neurochemical action of the vigilance-promoting drug modafinil.

  2000cites this paper
• Enhanced 5-HT metabolism and synthesis rate by the new selective r5-HT1B receptor antagonist, NAS-181 in the rat brain.

  2000cites this paper
• Characterization of endogenous serotonin-mediated regulation of dopamine release in the rat prefrontal cortex.

  1999cites this paper
• Chronic clomipramine and triiodothyronine increase serotonin levels in rat frontal cortex in vivo: relationship to serotonin autoreceptor activity.

  1999cites this paper
• Synergism between 5-HT1B/1D and 5-HT1A receptor antagonists on turnover and release of 5-HT in guinea-pig brain in vivo

  1999influential citation
• Diurnal variation in 5‐HT1B autoreceptor function in the anterior hypothalamus in vivo: effect of chronic antidepressant drug treatment

  1999cites this paper
• Differential effects of 5-HT1B/1D receptor antagonists in dorsal and median raphe innervated brain regions.

  1998cites this paper
• Role of Somatodendritic 5‐HT Autoreceptors in Modulating 5‐HT Neurotransmission a

  1998cites this paper
• Pharmacological analysis of G‐protein activation mediated by guinea‐pig recombinant 5‐HT1B receptors in C6‐glial cells: similarities with the human 5‐HT1B receptor

  1998cites this paper
• Possible serotonergic mechanisms underlying the antidepressant and anti-obsessive-compulsive disorder responses.

  1998cites this paper