Synthesis and evaluation of monoamidoxime derivatives: toward new antileishmanial compounds.

No abstract is available for this paper.

• Publication year

  2011

• Venue

  European journal of medicinal chemistry

• Publication date

  2011-07-01

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1016/j.ejmech.2011.04.026PMID 21555166
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Systematic review of the adverse effects of cutaneous leishmaniasis treatment in the New World.

  2011cited by this paper
• Synthesis and biological evaluation of L-valine-amidoximeesters as double prodrugs of amidines.

  2011cited by this paper
• Chemotherapy against human African trypanosomiasis: Is there a road to success?

  2010cited by this paper
• Theoretical models of pentamidine analogs activity based on their DNA minor groove complexes.

  2010cited by this paper
• Diamidines for human African trypanosomiasis.

  2010cited by this paper
• Synthesis and evaluation of original amidoximes as antileishmanial agents.

  2010cited by this paper
• In vitro activity of anti-leishmanial drugs against Leishmania donovani is host cell dependent.

  2010cited by this paper
• Coiled-coil conformation of a pentamidine-DNA complex.

  2010cited by this paper
• An efficient aqueous microwave-assisted Suzuki–Miyaura cross-coupling reaction in the thiazole series

  2009cited by this paper
• Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines.

  2009cited by this paper
• Microwave-assisted manganese(III) acetate based oxidative cyclizations of alkenes with β-ketosulfones

  2009cited by this paper
• Efficacy of the diamidine DB75 and its prodrug DB289, against murine models of human African trypanosomiasis.

  2008cited by this paper
• Pafuramidine for Pneumocystis jiroveci pneumonia in HIV-infected individuals

  2007cited by this paper
• Rapid synthesis of sulfone derivatives as potential anti-infectious agents.

  2007cited by this paper
• Visceral leishmaniasis: what are the needs for diagnosis, treatment and control?

  2007cited by this paper
• Bacterial pathogenesis: Clearing a path

  2007cited by this paper
• Dicationic DNA-targeted antiprotozoal agents: naphthalene replacement of benzimidazole.

  2006cited by this paper
• 5-Nitroimidazole Drugs Effective against Metronidazole-Resistant Trichomonas vaginalis and Giardia duodenalis

  2006cited by this paper
• Pentamidine uptake and resistance in pathogenic protozoa: past, present and future.

  2003cited by this paper
• Chemotherapy of human African trypanosomiasis: current and future prospects.

  2003cited by this paper
• 1,3-Diphenylpyrazoles: synthesis and antiparasitic activities of azomethine derivatives.

  2002cited by this paper
• Treatment and prophylaxis of Pneumocystis carinii pneumonia.

  1998cited by this paper
• Human leishmaniasis: clinical, diagnostic, and chemotherapeutic developments in the last 10 years.

  1997cited by this paper
• Synthesis and in vitro anti-protozoan activity of new 5-nitrothiophene oxime ether derivatives

  1993cited by this paper
• Genotoxicity in oxazolidine derivatives: influence of the nitro group

  1990cited by this paper
• Update on pentamidine for the treatment of Pneumocystis carinii pneumonia.

  1988cited by this paper
• Pentamidine: a review.

  1985cited by this paper
• Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays.

  1983cited by this paper

• Hit-to-lead optimization of 4,5-dihydrofuran-3-sulfonyl scaffold against Leishmania amazonensis. Effect of an aliphatic moiety.

  2024cites this paper
• Enhancing Antileishmanial Activity of Amidoxime-Based Compounds Bearing a 4,5-Dihydrofuran Scaffold: In Vitro Screening Against Leishmania amazonensis

  2024cites this paper
• Sonogashira Cross‐Coupling Reaction of Bromocyanofluoro Pyridine Compounds: Access to 5‐ and 6‐Alkynylfluoropyridinamidoximes Scaffolds

  2021cites this paper
• Optimization of the synthesis of het/aryl-amidoximes using an efficient green chemistry

  2020cites this paper
• Original antileishmanial hits: Variations around amidoximes.

  2018cites this paper
• Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series.

  2015cites this paper
• Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series.

  2015cites this paper
• New series of monoamidoxime derivatives displaying versatile antiparasitic activity.

  2014cites this paper
• Fruitful decade for antileishmanial compounds from 2002 to late 2011.

  2014cites this paper
• Synthesis and antileishmanial activity of novel pyridinium-hydrazone derivatives

  2013cites this paper
• Targeting the human parasite Leishmania donovani: discovery of a new promising anti-infectious pharmacophore in 3-nitroimidazo[1,2-a]pyridine series.

  2013cites this paper
• Manganese(III) Acetate-mediated Oxidative Cyclization of α-Methylstyrene and trans-Stilbene with β-Ketosulfones

  2013cites this paper
• A new, rapid and sensitive bioluminescence assay for drug screening on Leishmania.

  2013cites this paper
• Tandem synthesis and in vitro antiplasmodial evaluation of new naphtho[2,1-d]thiazole derivatives.

  2012cites this paper
• Cyclisations radicalaires oxydatives médiées par l'acétate de manganèse (III) et orientées vers la chimie médicinale

  2012cites this paper
• Access to original spirocyclic derivatives via inter- or intramolecular reaction mediated by manganese(III) acetate

  2012cites this paper
• New Methodology for the Synthesis of Thiobarbiturates Mediated by Manganese(III) Acetate

  2012cites this paper
• Preparation and antiprotozoal evaluation of promising β-carboline alkaloids.

  2012cites this paper
• Microwave and continuous flow technologies in drug discovery

  2012cites this paper
• Discovery of a new antileishmanial hit in 8-nitroquinoline series.

  2012cites this paper
• Nonneoplastic mucocutaneous lesions in organ transplant recipients

  2011cites this paper
• MAOS and Medicinal Chemistry: Some Important Examples from the Last Years

  2011cites this paper