Determination of neuropeptide Y Y1 receptor antagonist BIBP 3226 and evaluation of receptor expression based on liquid chromatography coupled with tandem mass spectrometry

No abstract is available for this paper.

• Publication year

  2020

• Venue

  Analytical and Bioanalytical Chemistry

• Publication date

  2020-07-29

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1007/s00216-020-02825-zPMID 32728863
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

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  1996cited by this paper
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  1994cited by this paper
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  1993cited by this paper
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