Phosphate and thiophosphate group donating adenine and guanine nucleotides inhibit glibenclamide binding to membranes from pancreatic islets

No abstract is available for this paper.

• Publication year

  2004

• Venue

  Naunyn-Schmiedeberg's Archives of Pharmacology

• Publication date

  Unknown publication date

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1007/BF00180681PMID 1903188
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Transphosphorylation and G protein activation.

  1990cited by this paper
• Tolbutamide-sensitivity of the adenosine 5′-triphosphate-dependent K+ channel in mouse pancreatic B-cells

  1990cited by this paper
• Protein phosphorylation is required for diazoxide to open ATP‐sensitive potassium channels in insulin (RINm5F) secreting cells

  1989cited by this paper
• Dual effects of diazoxide on ATP‐K+ currents recorded from an insulin‐secreting cell line

  1989cited by this paper
• Control of insulin secretion by sulfonylureas, meglitinide and diazoxide in relation to their binding to the sulfonylurea receptor in pancreatic islets.

  1989cited by this paper
• ATP-sensitive K-channels in HIT T15 β-cells studied by patch-clamp methods, 86Rb efflux and glibenclamide binding

  1989cited by this paper
• Adenosine 5'-triphosphate-sensitive potassium channels.

  1988cited by this paper
• Dual effects of ATP on K+ currents of mouse pancreatic β-cells

  1987cited by this paper
• Dual effects of ATP on K+ currents of mouse pancreatic beta-cells.

  1987cited by this paper
• G proteins: transducers of receptor-generated signals.

  1987cited by this paper
• Glucose-induced changes in cytosolic ATP content in pancreatic islets.

  1987cited by this paper
• Opposite effects of tolbutamide and diazoxide on the ATP-dependent K+ channel in mouse pancreatic β-cells

  1986cited by this paper
• A metabolite-regulated potassium channel in rat pancreatic B cells.

  1986cited by this paper
• Regulation of free and bound magnesium in rat hepatocytes and isolated mitochondria.

  1986cited by this paper
• ATP maintains ATP-inhibited K+ channels in an operational state

  1986cited by this paper
• The sulphonylurea receptor may be an ATP-sensitive potassium channel.

  1985cited by this paper
• Inhibition of 3H-glibenclamide binding to sulfonylurea receptors by oral antidiabetics.

  1985cited by this paper
• The enzymatic measurement of adenine nucleotides and P-creatine in picomole amounts.

  1981cited by this paper
• Some Statistical Methods Useful in Circulation Research

  1980cited by this paper
• Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction.

  1973cited by this paper
• [65] Assays of intermediates of the citric acid cycle and related compounds by fluorometric enzyme methods

  1969cited by this paper
• Pancreatic Islets in Mice with the Obese-hyperglycemic Syndrome: Lack of Effect of Carbutamide

  1960cited by this paper

• ATP binding without hydrolysis switches sulfonylurea receptor 1 (SUR1) to outward-facing conformations that activate KATP channels

  2018cites this paper
• Binding of sulphonylureas to plasma proteins – A KATP channel perspective

  2018cites this paper
• Neonatal Diabetes and Congenital Hyperinsulinism Caused by Mutations in ABCC8/SUR1 are Associated with Altered and Opposite Affinities for ATP and ADP

  2015cites this paper
• Sulfonylureas suppress the stimulatory action of Mg-nucleotides on Kir6.2/SUR1 but not Kir6.2/SUR2A KATP channels: A mechanistic study

  2014cites this paper
• Two Neonatal Diabetes Mutations on Transmembrane Helix 15 of SUR1 Increase Affinity for ATP and ADP at Nucleotide Binding Domain 2*

  2012cites this paper
• Some cannabinoid receptor ligands and their distomers are direct-acting openers of SUR1 K ATP channels

  2012cites this paper
• ABCC8: Physiology and Pathology*

  2011cites this paper
• Auswirkung des konservativen Aminosäurenaustauschs Lysin gegen Arginin in den Nukleotidbindungsfalten des Sulfonylharnstoffrezeptors SUR2B auf die Bindungsei- genschaften

  2010cites this paper
• Syntaxin-1A Inhibits the KATP Channel Through Interaction with Distinct Sites Along the Nucleotide-binding Folds of Sulfonylurea Receptor 1

  2010cites this paper
• Sulfonylurea receptors and mechanism of sulfonylurea action.

  2009cites this paper
• Incomplete dissociation of glibenclamide from wild‐type and mutant pancreatic KATP channels limits their recovery from inhibition

  2009cites this paper
• Chronic sustained and intermittent hypoxia reduce function of ATP-sensitive potassium channels in nucleus of the solitary tract.

  2008cites this paper
• Membrane ion channels and diabetes.

  2006cites this paper
• Lipids modulate ligand binding to sulphonylurea receptors

  2005influential citation
• Hydroxyl-substituted sulfonylureas as potent inhibitors of specific [3H]glyburide binding to rat brain synaptosomes.

  2003cites this paper
• Modulation of cardiac CaV1.2 channels by dihydropyridine and phosphatase inhibitor requires Ser-1142 in the domain III pore loop

  2003cites this paper
• The Stereoenantiomers of a Pinacidil Analog Open or Close Cloned ATP-sensitive K+ Channels*

  2002cites this paper
• Four novel splice variants of sulfonylurea receptor 1.

  2002cites this paper
• Sulfonylurea stimulation of insulin secretion.

  2002cites this paper
• Glibenclamide binding to sulphonylurea receptor subtypes: dependence on adenine nucleotides

  2002influential citation
• The common single nucleotide polymorphism E23K in K(IR)6.2 sensitizes pancreatic beta-cell ATP-sensitive potassium channels toward activation through nucleoside diphosphates.

  2002cites this paper
• Interaction of K(ATP) channel modulators with sulfonylurea receptor SUR2B: implication for tetramer formation and allosteric coupling of subunits.

  2002cites this paper
• Modulation by Nucleotides of Binding Sites for [3H]Glibenclamide in Rat Aorta and Cardiac Ventricular Membranes

  2001cites this paper
• Changes in [(3)H]glibenclamide binding to mouse forebrain membranes during morphine tolerance.

  2001cites this paper
• The beta-cell K(ATP) channel.

  2000cites this paper
• Stoichiometry of sulfonylurea-induced ATP-sensitive potassium channel closure.

  1999cites this paper
• The tolbutamide site of SUR1 and a mechanism for its functional coupling to KATP channel closure

  1999cites this paper
• Identification of the Potassium Channel Opener Site on Sulfonylurea Receptors*

  1999cites this paper
• Potassium channel openers require ATP to bind to and act through sulfonylurea receptors

  1998cites this paper
• Evidence for a 65 kDa sulfonylurea receptor in rat pancreatic zymogen granule membranes

  1997cites this paper
• Evidence for a Unique Long Chain Acyl-CoA Ester Binding Site on the ATP-regulated Potassium Channel in Mouse Pancreatic Beta Cells*

  1997cites this paper
• Sulphonylurea binding in rat isolated glomeruli: pharmacological characterization and dependence on cell metabolism and cytoskeleton

  1997cites this paper
• Developmental and tissue-specific sulfonylurea receptor gene expression.

  1997cites this paper
• Effects of protein phosphorylation on the sulphonylurea receptor of the pancreatic beta-cell.

  1997cites this paper
• Putative pre- and postsynaptic ATP-sensitive potassium channels in the rat substantia nigra in vitro

  1995cites this paper
• Interaction of fluorescein derivatives with sulfonylurea binding in insulin-secreting cells.

  1995cites this paper
• Cloning of the beta cell high-affinity sulfonylurea receptor: a regulator of insulin secretion.

  1995cites this paper
• Interaction of tolbutamide and cytosolic nucleotides in controlling the ATP‐sensitive K+ channel in mouse β‐cells

  1994cites this paper
• KATP--fact or artefact? New thoughts on the mode of action of the potassium channel openers.

  1994cites this paper
• Mg(2+)-dependent inhibition of KATP by sulphonylureas in CRI-G1 insulin-secreting cells.

  1994cites this paper
• Photoaffinity Labeling of the Cerebral Sulfonylurea Receptor Using a Novel Radioiodinated Azidoglibenclamide Analogue

  1994cites this paper
• Protein phosphorylation and beta-cell function

  1994cites this paper
• Antagonism of the stimulatory effects of efaroxan and glibenclamide in rat pancreatic islets by the imidazoline, RX801080

  1993cites this paper
• The pharmacology of ATP-sensitive potassium channels.

  1993cites this paper
• Sulfonylurea-binding sites and ATP-sensitive K+ channels in alpha-TC glucagonoma and beta-TC insulinoma cells.

  1993cites this paper
• Nucleotides modulate the low affinity binding sites for [3H]glibenclamide in the rat brain.

  1993cites this paper
• Regional distribution of sulfonylurea receptors in the brain of rodent and primate.

  1993cites this paper
• Antagonism of levcromakalim by imidazoline‐ and guanidine‐derivatives in rat portal vein: involvement of the delayed rectifier

  1993cites this paper
• Levcromakalim may induce a voltage‐independent K‐current in rat portal veins by modifying the gating properties of the delayed rectifier

  1993cites this paper
• Induction of a glibenclamide‐sensitive K‐current by modification of a delayed rectifier channel in rat portal vein and insulinoma cells

  1993cites this paper
• The beta-cell sulfonylurea receptor.

  1993cites this paper
• Mg2+ modulates the binding of [3H]glibenclamide to its receptor in rat cerebral cortical membranes.

  1993cites this paper
• Evidence for a saturable, energy-dependent and carrier-mediated uptake of oral antidiabetics into rat hepatocytes.

  1992cites this paper
• Adenine nucleotide‐induced inhibition of binding of sulphonylureas to their receptor in pancreatic islets

  1992cites this paper
• Diazoxide‐sensitivity of the adenosine 5′‐triphosphate‐dependent K+ channel in mouse pancreatic β‐cells

  1992cites this paper
• Pancreatic and Extrapancreatic Sulfonylurea Receptors

  1992cites this paper
• The sulfonylurea receptor.

  1992cites this paper
• The binding properties of the solubilized sulfonylurea receptor from a pancreatic B-cell line are modulated by the Mg(++)-complex of ATP.

  1992cites this paper
• The Binding Properties of the Particulate and Solubilized Sulfonylurea Receptor from Cerebral Cortex Are Modulated by the Mg2+ Complex of ATP

  1992cites this paper
• Inhibition of energy metabolism by 3-nitropropionic acid activates ATP-sensitive potassium channels.

  1992cites this paper
• Effects of pH upon the inhibition by sulphonylurea drugs of ATP-sensitive K+ channels in cardiac muscle.

  1992cites this paper
• Potassium channels of the insulin‐secreting B cell

  1992cites this paper
• Cytosolic nucleotides enhance the tolbutamide sensitivity of the ATP-dependent K+ channel in mouse pancreatic B cells by their combined actions at inhibitory and stimulatory receptors.

  1992cites this paper
• Effect of MgATP on pinacidil‐induced displacement of glibenclamide from the sulphonylurea receptor in a pancreatic β‐cell line and rat cerebral cortex

  1992cites this paper
• Chronic Sustained and Intermittent Hypoxia Reduce the Function of Atp-sensitive Potassium Channels in the Nucleus of the Solitary Tract

  year unknowncites this paper