Short Communication New 5‐HT1A receptor antagonist: [3H]p‐MPPF

No abstract is available for this paper.

• Publication year

  1996

• Venue

  Synapse

• Publication date

  1996-08-01

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1002/(SICI)1098-2396(199608)23:4<344::AID-SYN13>3.0.CO;2-XPMID 8855520
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

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  1995cited by this paper
• Quantitative autoradiographic characterisation of the binding of [3H]WAY-100635, a selective 5-HT1A receptor antagonist.

  1995cited by this paper
• The selective 5-HT1A antagonist radioligand [3H]WAY 100635 labels both G-protein-coupled and free 5-HT1A receptors in rat brain membranes.

  1995cited by this paper
• Synthesis and evaluation of 4-(2'-methoxyphenyl)-1-[2'-[N-(2"-pyridinyl)-p- iodobenzamido]ethyl]piperazine (p-MPPI): a new iodinated 5-HT1A ligand.

  1994cited by this paper
• International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (Serotonin).

  1994cited by this paper
• Silent 5-HT1A receptor antagonists: utility as research tools and therapeutic agents.

  1993cited by this paper
• The putative 5-HT1A receptor antagonists NAN-190 and BMY 7378 are partial agonists in the rat dorsal raphe nucleus in vitro.

  1992cited by this paper
• Serotonin receptors and their ligands: a lack of selective agents.

  1991cited by this paper
• Species differences in the distribution of central 5-HT1 binding sites: a comparative autoradiographic study between rat and guinea pig.

  1991cited by this paper
• Analogues of the 5-HT1A serotonin antagonist 1-(2-methoxyphenyl)-4-[4-(2-phthalimido)butyl]piperazine with reduced alpha 1-adrenergic affinity.

  1991cited by this paper
• NAN-190: agonist and antagonist interactions with brain 5-HT1A receptors.

  1990cited by this paper
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  1990cited by this paper
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  1988cited by this paper
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  1988cited by this paper

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• Neurotransmission sérotoninergique 5-HT1A : approche méthodologique de la mesure in vivo par le [18F]MPPF en tomographie par émission de positons

  2007cites this paper
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  2007cites this paper
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  2007cites this paper
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  2006cites this paper
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  2006cites this paper
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  2006cites this paper
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• PET Studies on P-glycoprotein function in the blood-brain barrier: how it affects uptake and binding of drugs within the CNS.

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  2003cites this paper
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  2002cites this paper
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