Synthesis, antiproliferative activity and genotoxicity of novel anthracene-containing aminophosphonates and a new anthracene-derived Schiff base.

No abstract is available for this paper.

• Publication year

  2012

• Venue

  Bioorganic & Medicinal Chemistry

• Publication date

  Unknown publication date

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1016/j.bmc.2011.11.024PMID 22142614
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Phenylimino-10H-anthracen-9-ones as novel antimicrotubule agents-synthesis, antiproliferative activity and inhibition of tubulin polymerization.

  2011cited by this paper
• Research Article: Asymmetric Hydrophosphylation of Chiral N‐Phosphonyl Imines Provides an Efficient Approach to Chiral α‐Amino Phosphonates

  2010cited by this paper
• Aminophosphonic acids and derivatives. Synthesis and biological applications.

  2010cited by this paper
• Synthesis, antiproliferative activity and inhibition of tubulin polymerization by 1,5- and 1,8-disubstituted 10H-anthracen-9-ones bearing a 10-benzylidene or 10-(2-oxo-2-phenylethylidene) moiety.

  2010cited by this paper
• 10-(2-oxo-2-phenylethylidene)-10H-anthracen-9-ones as highly active antimicrotubule agents: synthesis, antiproliferative activity, and inhibition of tubulin polymerization.

  2009cited by this paper
• A new strategy for asymmetric synthesis of aminophosphonic acid derivatives: the first enantioselective catalytic reduction of C-phosphorylated imines

  2009cited by this paper
• An Overview of Stereoselective Synthesis of α-Aminophosphonic Acids and Derivatives.

  2009cited by this paper
• Irreversible inhibition of serine proteases - design and in vivo activity of diaryl alpha-aminophosphonate derivatives.

  2009cited by this paper
• Targeting Enzymes with Phosphonate-Based Inhibitors: Mimics of Tetrahedral Transition States and Stable Isosteric Analogues of Phosphates

  2006cited by this paper
• The search of DNA-intercalators as antitumoral drugs: what it worked and what did not work.

  2005cited by this paper
• Novel benzylidene-9(10H)-anthracenones as highly active antimicrotubule agents. Synthesis, antiproliferative activity, and inhibition of tubulin polymerization.

  2003cited by this paper
• Synthesis and NMR Spectroscopic Study of a New Anthracene Derived Schiff Base and a Bis(aminophosphonate) Obtained from It

  2003cited by this paper
• An Overview of Recent Advances on the Synthesis and Biological Activity of α‐Aminophosphonic Acid Derivatives

  2001cited by this paper
• Physiological Activity of Some Organophosphorous Compounds and Their Influence on Mechanical Properties of Erythrocytes

  2001cited by this paper
• Biodistribution and Pharmacokinetics of Variously Sized Molecular Radiolabelled Polyethyleneiminomethyl Phosphonic Acid as a Selective Bone Seeker for Therapy in the Normal Primate Model

  2001cited by this paper
• Syntheses, characterization, stereochemistry and complexing properties of acyclic and macrocyclic compounds possessing α‐amino‐ or α‐hydroxyphosphonate units: a review article

  2000cited by this paper
• Aminophosphonic and aminophosphinic acids : chemistry and biological activity

  2000cited by this paper
• Synthesis of 1,4-phenylene-bis-aminomethanephosphonates: The stereochemical aspect

  2000cited by this paper
• [Placebo effects and adverse effects in clinical trials].

  2000cited by this paper
• The International EU/COLIPA In Vitro Phototoxicity Validation Study: Results of Phase II (Blind Trial). Part 1: The 3T3 NRU Phototoxicity Test.

  1998cited by this paper
• Structure-Activity Studies of Aminophosphonic Derivatives of Fluorene

  1996cited by this paper
• Peptide synthesis catalyzed by an antibody containing a binding site for variable amino acids.

  1994cited by this paper
• Mammalian in vivo cytogenetic assays. Analysis of chromosome aberrations in bone marrow cells.

  1987cited by this paper
• Comparative molecular pharmacology in leukemic L1210 cells of the anthracene anticancer drugs mitoxantrone and bisantrene.

  1985cited by this paper
• Toxicity determined in vitro by morphological alterations and neutral red absorption.

  1985cited by this paper
• Anthracenyl crown ethers and cryptands as fluorescent probes for solid-phase transitions of phosphatidylcholines: syntheses and phospholipid membrane studies.

  1984cited by this paper
• Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays.

  1983cited by this paper
• 13C NMR of polycyclic aromatic compounds. A review

  1979cited by this paper
• 13C n.m.r. spectroscopy of diethyl alkyl- and benzyl-phosphonates. A study of phosphorus–carbon spin–spin coupling constants over one to seven bonds

  1977cited by this paper

• Cytotoxicity and structural manipulations of biomimetic salicylidene based compounds

  2025cites this paper
• Pharmacological Activities of Schiff Bases and Their Derivatives with Low and High Molecular Phosphonates

  2023cites this paper
• Niobium Pentachloride Mediated Direct Bradsher-Type Reaction: A Rapid and Efficient Strategy to Synthesize Novel Substituted 9-Anthraldehydes

  2023cites this paper
• Antioxidant and cytotoxic activities of selected salicylidene imines: experimental and computational study

  2022influential citation
• A new bio-active asymmetric-Schiff base: synthesis and evaluation of calf thymus DNA interaction, topoisomerase IIα inhibition, in vitro antiproliferative activity, SEM analysis and molecular docking studies

  2022cites this paper
• Theoretical exploration on structures, bonding aspects and molecular docking of α-aminophosphonate ligated copper complexes against SARS-CoV-2 proteases

  2022cites this paper
• Schiff Bases: Interesting Scaffolds with Promising Antitumoral Properties

  2021influential citation
• Anthracene‐Based Triazolyl Triethoxysilanes as Selective and Colorimetric Sensor for Cysteine: Rationalization towards Stability Factors, Therapeutics Evaluation and Molecular Docking

  2021cites this paper
• Copper (II) complexes derived from pyridoxal: Structural correlations, cytotoxic activities, and molecular docking

  2021cites this paper
• New Mn(II) and Cu(II) Complexes of Naphtaldimine Schiff Base Ligands: Synthesis, Characterization and Crystal Structures

  2020cites this paper
• Rosmarinic acid prevents gastric ulcers via sulfhydryl groups reinforcement, antioxidant and immunomodulatory effects

  2020cites this paper
• Synthesis, molecular structure and antioxidant activity of bis [L(μ2-chloro)copper(II)] supported by phenoxy/naphthoxy-imine ligands.

  2020cites this paper
• Synthesis of novel α-aminophosphonates under microwave irradiation, biological evaluation as antiproliferative agents and apoptosis inducers

  2019cites this paper
• Design, Synthesis and Structural Inspection of Some Novel Di- And Tri-Azomethene Compounds as Chemo Sensors for the Detection of Various Metal Ions

  2019cites this paper
• Reactivity of P–H Group of H-Phosphinic Acid and Its Derivatives

  2018cites this paper
• Synthesis of Two Novel Homologous Polyphosphoesters Containing Aminophosphonate Units and Cytotoxicity of Some Low-Molecular and Polymeric Aminophosphonate Derivatives

  2018cites this paper
• Synthesis of fluorescent aminophosphonates by green chemistry procedures

  2017cites this paper
• Promiscuous lipase catalyzed a new P–C bond formation: Green and efficient protocol for one‐pot synthesis of α‐aminophosphonates

  2017cites this paper
• The synthesis of α-aryl-α-aminophosphonates and α-aryl-α-aminophosphine oxides by the microwave-assisted Pudovik reaction

  2017cites this paper
• Microwave assisted synthesis and X-ray structure of a novel anthracene-derived aminophosphonate. Enantioseparation of two α-aminophosphonates and genotoxicity in vivo

  2017cites this paper
• Convenient Synthesis of Cyclic α‐Aminophosphonates by Alkylation–Cyclization Reaction of Iminophosphoglycinates Using Phase‐Transfer Catalysis

  2016cites this paper
• In vitro antitumour activity, safety testing and subcellular distribution of two poly[oxyethylene(aminophosphonate-co-H-phosphonate)]s in Ehrlich ascites carcinoma and BALB/c 3T3 cell culture systems

  2016cites this paper
• Synthesis, antiproliferative and apoptosis-inducing effects of novel asiatic acid derivatives containing α-aminophosphonates

  2016cites this paper
• Rapid Access to New Thiazepinyl and Oxazepinyl Phosphonates through a Green Pudovik Reaction

  2016cites this paper
• 4. Synthesis of Organophosphines, Phosphonates, and Related Compounds

  2016cites this paper
• Novel symmetric diimine-Schiff bases and asymmetric triimine-Schiff bases as chemosensors for the detection of various metal ions

  2016cites this paper
• EXPLORING NOVEL HETEROCYCLICS - AN INSIGHT TO SYNTHETIC STRATEGY AND BIOLOGICAL ACTIVITY.

  2015cites this paper
• Mutagenic assessment of three synthetic pyridine-diaryl ketone derivatives

  2015cites this paper
• An update on the stereoselective synthesis of α-aminophosphonic acids and derivatives

  2015cites this paper
• Comparative assessment of in vitro and in vivo biological activity of some anthracene-derived aminophosphonates , bis-aminophosphonates and poly ( aminophosphonate ) s

  2014cites this paper
• Synthesis, characterization, antitumor activity and safety testing of novel polyphosphoesters bearing anthracene-derived aminophosphonate units.

  2014cites this paper
• 3 COMPARATIVE ASSESMENT OF IN VITRO AND IN VIVO BIOLOGICAL ACTIVITY OF SOME RECENTLY SYNTHESIZED AMINOPHOSPHONATES , BIS-AMINOPHOSPHONATES AND POLY ( AMINOPHOSPHONATE )

  2014cites this paper
• Quality evaluation of semen oroxyli based on the determination of multiple components with a single reference standard.

  2013cites this paper
• Synthesis of Biologically Active α-Aminophosphonates

  2013cites this paper
• Anthracene-Derived Bis-Aminophosphonates: Crystal Structure, In Vitro Antitumor Activity, and Genotoxicity In Vivo

  2013cites this paper
• An insight into synthetic Schiff bases revealing antiproliferative activities in vitro.

  2013cites this paper
• Synthesis, Structural Elucidation, and In Vitro Antitumor Activities of Some Pyrazolopyrimidines and Schiff Bases Derived from 5-Amino-3-(arylamino)-1H-pyrazole-4-carboxamides

  2013cites this paper
• Synthesis and NMR Characterization of Two Novel Anthracene-Derived BIS-Aminophosphonates. Basic Hydrolysis of Some Aminophosphonate Derivatives

  2012cites this paper
• Diethyl [(9-anthryl)(4-methylanilino)methyl]phosphonate

  2011cites this paper
• rac-Dimethyl [(9-anthryl)(4-methylanilino)methyl]phosphonate

  2011cites this paper
• COMPARATIve sTUDy BeTweeN TOxIC e��eCTs O� Newly syNTHesIZeD AMINOPHOsPHATes (AP) AND glyPHOsATe ON �ResH-wATeR CIlIATes MODel; ParameCium tetraurelia

  year unknowncites this paper