Pharmacological profile of a novel class of muscarinic acetylcholine receptor agonists.

No abstract is available for this paper.

• Publication year

  1986

• Venue

  European Journal of Pharmacology

• Publication date

  1986-10-14

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1016/0014-2999(86)90191-3PMID 3780854
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• The specific protective effect of diazepam and valproate against isoniazid-induced seizures is not correlated with increased GABA levels

  2005cited by this paper
• Prodrugs as drug delivery systems. 43. O-acyloxymethyl salicylamide N-Mannich bases as double prodrug forms for amines

  1986cited by this paper
• Changes in Nicotinic and Muscarinic Cholinergic Receptors in Alzheimer‐Type Dementia

  1986cited by this paper
• A novel class of conformationally restricted heterocyclic muscarinic agonists.

  1986cited by this paper
• Decreased Muscarinic Acetylcholine Receptor Number in the Central Nervous System of the Tottering (tg/tg) Mouse

  1986cited by this paper
• Neurochemistry of aging. 1. Toxins for an animal model of Alzheimer's disease.

  1986cited by this paper
• Knife cuts of entorhinal cortex: effects on development of amygdaloid kindling and seizure-induced decrease of muscarinic cholinergic receptors

  1985cited by this paper
• Cholinergic Drugs and Memory

  1985cited by this paper
• Role of neurotransmitters in seizure mechanisms in the kindling model of epilepsy.

  1984cited by this paper
• Choline acetyltransferase immunohistochemistry in brains of Alzheimer's disease patients and controls.

  1983cited by this paper
• Chemical kindling by muscarinic amygdaloid stimulation in the rat.

  1983cited by this paper
• The substantia innominata in Alzheimer's disease: an histochemical and biochemical study of cholinergic marker enzymes.

  1982cited by this paper
• Antinociceptive and anticonvulsive effect of THIP, a pure GABA agonist.

  1982cited by this paper
• The cholinergic hypothesis of geriatric memory dysfunction.

  1982cited by this paper
• Cortical muscarinic receptor subtypes and Alzheimer's disease.

  1982cited by this paper
• Physostigmine and Arecoline: Effects of Intravenous Infusions in Alzheimer Presenile Dementia

  1981cited by this paper
• A comparison of muscarinic cholinergic involvement in the antinociceptive effects of morphine and clonidine in the mouse.

  1980cited by this paper
• The central action of various arecaidine esters (arecoline derivatives) on blood pressure and heart rate in the cat. Comparison with the peripheral effects.

  1978cited by this paper
• Morphine‐like ligand for opiate receptors in human CSF

  1975cited by this paper
• Partition coefficients and their uses

  1971cited by this paper
• Narcotic-antagonist analgesics: interactions with cholinergic systems.

  1969cited by this paper
• [On the pharmacology of active materials from betel. 2. Transformation of arecoline to arecaidine].

  1968cited by this paper
• pAx and competitive drug antagonism.

  1949cited by this paper

• Green Chemistry Approach to Fast and Highly Efficient One-Pot Synthesis of Bis-Isoxazolyl-1,2,5,6-Tetrahydro Pyridine-3-Carboxylates

  2013cites this paper
• Betel Quid and Areca Nut

  2012cites this paper
• Selective muscarinic ligands (a review)

  2004cites this paper
• Synthesis and muscarinic receptor pharmacology of a series of 4,5,6,7-tetrahydroisothiazolo[4,5-c]pyridine bioisosteres of arecoline.

  1999cites this paper
• In vivo muscarinic cholinergic mediated effects of Lu 25-109, a M1 agonist and M2/M3 antagonist in vitro

  1998cites this paper
• 3-(3-Alkylthio- 1,2,5-thiadiazol-4-yl)- 1 -azabicycles. Structure-activity relationships for antinociception mediated by central muscarinic receptors

  1996cites this paper
• Annulated heterocyclic bioisosteres of norarecoline. Synthesis and molecular pharmacology at five recombinant human muscarinic acetylcholine receptors.

  1995cites this paper
• Muscarinic agonists as analgesics. Antinociceptive activity versus M1 activity: SAR of alkylthio-TZTP's and related 1,2,5-thiadiazole analogs.

  1995cites this paper
• The mouse grid-shock analgesia test: pharmacological characterization of latency to vocalization threshold as an index of antinociception.

  1994cites this paper
• Modification of the duration of action and pharmacodynamics of arecoline by tetraisopropylpyrophosphoramide.

  1994cites this paper
• The Muscarinic Receptors

  1989cites this paper
• Structural Determinants of Muscarinic Agonist Activity

  1989cites this paper
• Cognition activators

  1988cites this paper
• Heterocyclic muscarinic agonists. Synthesis and biological activity of some bicyclic sulfonium arecoline bioisosteres.

  1988cites this paper
• Chapter 4. Agents for the Treatment of Cognitive Disorders

  1988cites this paper