Benzodiazepines compete for thyrotropin-releasing hormone receptor binding: micromolar potency in rat pituitary, retina and amygdala.

No abstract is available for this paper.

• Publication year

  1983

• Venue

  Neuroscience Letters

• Publication date

  1983-11-11

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1016/0304-3940(83)90467-6PMID 6320064
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Biochemical similarity of rat pituitary and CNS TRH receptors.

  1983cited by this paper
• Receptors for thyrotropin-releasing hormone (TRH) in rabbit spinal cord.

  1983cited by this paper
• Benzodiazepine receptors in the central nervous system.

  1982cited by this paper
• Regulatory peptides as a source of new drugs--the clinical prospects for analogues of TRH which are resistant to metabolic degradation.

  1982cited by this paper
• Benzodiazepine receptors in the central nervous system.

  1982cited by this paper
• Micromolar affinity benzodiazepine receptors: identification and characterization in central nervous system.

  1982cited by this paper
• Effects of TRH on central nervous system function.

  1981cited by this paper
• Thyrotropin-releasing hormone improves cardiovascular function in experimental endotoxic and hemorrhagic shock.

  1981cited by this paper
• Binding sites for thyrotropin-releasing hormone in sheep nucleus accumbens resemble pituitary receptors.

  1980cited by this paper
• Effect of thyrotropin-releasing hormone on ataxia of spinocerebellar degeneration.

  1980cited by this paper
• Attenuation of the effect of punishment by thyrotropin-releasing hormone: comparisons with chlordiazepoxide.

  1980cited by this paper
• Problems Associated with the Binding of L‐Glutamic Acid to Synaptic Membranes: Methodological Aspects

  1980cited by this paper
• Multiple serotonin receptors: differential binding of [3H]5-hydroxytryptamine, [3H]lysergic acid diethylamide and [3H]spiroperidol.

  1979cited by this paper
• The binding of antagonists to brain muscarinic receptors.

  1978cited by this paper
• The binding of agonists to brain muscarinic receptors.

  1978cited by this paper
• Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.

  1977cited by this paper
• 3H-Spiroperidol labels dopamine receptors in pituitary and brain.

  1977cited by this paper
• Beta adrenergic receptor binding in membrane preparations from mammalian brain.

  1976cited by this paper
• Letter: Insulin extraction and hepatic blood-flow.

  1976cited by this paper
• Opiate receptor mechanisms.

  1975cited by this paper
• Effects of thyrotropin-releasing hormone (TRH) on the actions of pentobarbital and other centrally acting drugs.

  1975cited by this paper
• Benzodiazepines in Clinical Practice

  1974cited by this paper
• Relationships between inhibition constants and fractional inhibition in enzyme-catalyzed reactions with different numbers of reactants, different reaction mechanisms, and different types and mechanisms of inhibition.

  1974cited by this paper
• Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction.

  1973cited by this paper
• THR (lopremone): psychobiological responses of normal women. I. Subjective experiences.

  1973cited by this paper

• Paradoxical GH response to TRH during status epilepticus in man.

  1999cites this paper
• Pilot investigation of thyrotropin-releasing hormone-induced thyrotropin and prolactin release in anxious patients treated with diazepam.

  1998cites this paper
• Involvement of glutamate and gamma-aminobutyric acid (GABA)-ergic systems in thyrotropin-releasing hormone-induced rat cerebellar cGMP formation.

  1996cites this paper
• Identification of thyrotropin-releasing hormone receptor in the rat testis.

  1994cites this paper
• Growth hormone response to growth hormone-releasing hormone in early abstinent alcoholic patients.

  1993cites this paper
• Peripheral-Type Mitochondrial Binding Sites for Benzodiazepines in GH3 Pituitary Cells

  1992cites this paper
• Thyrotropin-releasing hormone selectively reverses lorazepam-induced sedation but not slowing of saccadic eye movements.

  1992cites this paper
• Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.

  1992cites this paper
• Regional changes in central nervous system thyrotropin-releasing hormone after pentylenetetrazol-induced seizures in dogs.

  1992cites this paper
• Atipamezole, benzodiazepines, bicucullin and tifluadom antagonize the effect of TRH on rat duodenum and displace it from brain and anterior pituitary receptors.

  1991cites this paper
• Administration of chlordiazepoxide affects [3H][3-MeHis2]thyrotropin-releasing hormone binding in rat brain.

  1991cites this paper
• Central and peripheral type benzodiazepine ligands displace [3H][3-ME-HIS2]TRH from its binding sites in the brain and the anterior pituitary and antagonize the effect of TRH in the rat duodenum.

  1991cites this paper
• Effects of intra-amygdalar thyrotropin releasing hormone (TRH) and its antagonism by atropine and benzodiazepines during stress ulcer formation in rats.

  1990cites this paper
• Pharmacological and biochemical comparison of thyrotropin releasing hormone (TRH) and di‐methyl proline‐TRH on pituitary GH3 cells

  1990cites this paper
• Role of TRH in Seizure Modulation a

  1989cites this paper
• Mechanistic and functional divergence between thyrotropin-releasing hormone and RO 15-4513 interactions with ethanol.

  1989cites this paper
• The interaction of benzodiazepines with thyrotropin‐releasing hormone receptors on clonal pituitary cells

  1989cites this paper
• Use of Receptor Antagonists in Elucidating the Mechanism of Action of TRH in GH3 Cells a

  1989cites this paper
• Benzodiazepines modulate voltage-sensitive calcium channels in GH3 pituitary cells at sites distinct from thyrotropin-releasing hormone receptors.

  1988cites this paper
• Inhibition of the binding and the behavioral effects of thyrotropin-releasing hormone (TRH) by the triazolobenzodiazepines.

  1988cites this paper
• Autoradiographic localization of thyr tropin releasing hormone receptors in human brain

  1986cites this paper
• Benzodiazepine interactions with central thyroid-releasing hormone binding sites: characterization and physiological significance.

  1986cites this paper
• Evidence for tight coupling of receptor occupancy by thyrotropin-releasing hormone to phospholipase C-mediated phosphoinositide hydrolysis in rat pituitary cells: use of chlordiazepoxide as a competitive antagonist.

  1986cites this paper
• Benzodiazepines inhibit thyrotropin (TSH)-releasing hormone-induced TSH and growth hormone release from perifused rat pituitaries.

  1986cites this paper
• Evidence for a role of central type benzodiazepine receptors in the inhibition of the thyrotropin-releasing hormone-induced thyrotropin release from rat perifused pituitaries.

  1986cites this paper
• Thyrotropin-releasing hormone receptors in gut tissues resemble pituitary receptors.

  1986cites this paper
• Pharmacology of thyrotropin-releasing hormone.

  1986cites this paper
• THYROTROPIN-RELE ASING HORMONE

  1986cites this paper
• Ibotenic acid decreases thyrotropin-releasing hormone receptor binding in the rat amygdala.

  1985cites this paper
• Thyrotrophin releasing hormone: endocrine and central effects.

  1985cites this paper
• Chlordiazepoxide is a competitive thyrotropin-releasing hormone receptor antagonist in GH3 pituitary tumour cells.

  1985cites this paper
• Visualization and identification of TRH receptors in rodent brain by autoradiography and radioreceptor assays: focus on amygdala, N. accumbens, septum and cortex.

  1985cites this paper
• [Concentration of regulatory peptides in the cerebral cortex and their central activity].

  1985cites this paper
• Thyrotropin‐Releasing Hormone Receptor Binding Sites: Autoradiographic Distribution in the Rat and Guinea Pig Brain

  1985cites this paper
• Modulation of Receptors for Thyrotropin‐Releasing Hormone by Benzodiazepines: Brain Regional Differences

  1984cites this paper
• PITUITARY AND CNS TRH RECEPTORS

  1984cites this paper