B. Biersack

New N-Heterocyclic Carbene Gold and Platinum Complexes with 1,3-Dialkyl-4-anisyl-5-(4-chlorophenyl)imidazol-2-ylidene Ligands for the Treatment of Esophageal Adenocarcinoma.
20260 citationsauthor #7
Tuning the Dielectric Properties of Individual Clay Nanosheets by Interlayer Composition: Toward Nano‐Electret Materials
20251 citationsauthor #4
Curcumin and Its Derivatives in Hepatology: Therapeutic Potential and Advances in Nanoparticle Formulations
20257 citationsauthor #5
Identification of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Inhibitors Based on 2-Hydroxy-1,4-naphthoquinone Mannich Bases
20254 citationsauthor #10
A drug-repurposing screen of FDA- and EMA-approved drugs identifies two NF-κB inhibitors active against eumycetoma
20251 citationsauthor #3
Antiparasitic Evaluation and In Silico Investigation of New Acyl Hydrazones from 3-Iodo-5-methoxy-4-propargyloxybenzaldehyde
20250 citationsauthor #8
Kinome analysis of Madurella mycetomatis identified kinases in the cell wall integrity pathway as novel potential therapeutic drug targets in eumycetoma caused by Madurella mycetomatis
20250 citationsauthor #12
Abstract 6927: Novel ferrocene and naphthalene-based analogs block HRH1-signaling to inhibit colon cancer growth
20251 citationsauthor #6
Special Issue “Antifungal Drug Discovery: Progresses, Challenges, Opportunities”
20251 citationsauthor #1
Histone deacetylases in the regulation of cell death and survival mechanisms in resistant BRAF-mutant cancers
20252 citationsauthor #1
Antiparasitic and Antifungal Activities of Cetyl-Maritima, a New N-Cetyl-Modified Maritima Derivative
20250 citationsauthor #8
Collaborative Synthesis for Neglected Diseases through the Open Synthesis Network: Structure–Activity Relationships of Arylaminopyrazoles as Chagas Disease Treatments
20250 citationsauthor #72
Effects of Tyrphostin A9 and Structurally Related Tyrphostins on Colorectal Carcinoma Cells
20250 citationsauthor #8
In Vitro and In Silico Evaluation of the Anticancer and Antiparasitic Activities of New 2‐Methoxy Azachalconium Bromides
20250 citationsauthor #10
Exploring a Therapeutic Gold Mine: The Antifungal Potential of the Gold-Based Antirheumatic Drug Auranofin
20254 citationsauthor #3
Design, Hemisynthesis, Characterization, Molecular Docking, and Dynamics Evaluation of Novel Totarol‐1,2,3‐Triazole Derivatives as Leishmaniasis and Toxoplasmosis Agents
20252 citationsauthor #12
Identification of a New Pentafluorosulfanyl-Substituted Chalcone with Activity Against Hepatoma and Human Parasites
20250 citationsauthor #9
Role and Function of Receptor Tyrosine Kinases in BRAF Mutant Cancers
20249 citationsauthor #1
The Antifungal Potential of Niclosamide and Structurally Related Salicylanilides
202412 citationsauthor #1
Antimetastatic activity of (arene)ruthenium(II) complex of 4-aryl-4H-naphthopyran.
20242 citationsauthor #4
Emerging role of MYB transcription factors in cancer drug resistance
20246 citationsauthor #1
The influence of substituted indigo derivatives on the preparation and properties of ´´Maya´´ pigments
20240 citationsauthor #14
Antiparasitic Activities of Acyl Hydrazones from Cinnamaldehydes and Structurally Related Fragrances
20243 citationsauthor #5
Superior Anticancer and Antifungal Activities of New Sulfanyl-Substituted Niclosamide Derivatives
20243 citationsauthor #10
Therapeutic Potential of Aryl Sulfonamides: Synthesis, Antiproliferative, Antioxidant, Antiparasitic and Molecular Docking Studies
20241 citationsauthor #12
Antifungal Activity of Natural Naphthoquinones and Anthraquinones against Madurella mycetomatis
20238 citationsauthor #4
Regiospecific Reduction of 4,6‐Dinitrobenzimidazoles: Synthesis, Characterization, and Biological Evaluation
20233 citationsauthor #12
Synthetic Small Molecule Modulators of Hsp70 and Hsp40 Chaperones as Promising Anticancer Agents
202316 citationsauthor #3
Analogs of the Catechol Derivative Dynasore Inhibit HIV-1 Ribonuclease H, SARS-CoV-2 nsp14 Exoribonuclease, and Virus Replication
20237 citationsauthor #11
Abstract 1585: Targeting acid ceramidase-1 to inhibit sphingolipid metabolism and tumor growth in pancreatic ductal carcinoma
20231 citationsauthor #10
New Functional Polymer Materials via Click Chemistry-Based Modification of Cellulose Acetate
202310 citationsauthor #13
Synthesis, Physicochemical Characterization using a Facile Validated HPLC Quantitation Analysis Method of 4-Chloro-phenylcarbamoyl-methyl Ciprofloxacin and Its Biological Investigations
202321 citationsauthor #1
Synthesis and Anticancer Evaluation of New Indole-Based Tyrphostin Derivatives and Their (p-Cymene)dichloridoruthenium(II) Complexes
202311 citationsauthor #7
Multimodal 4-arylchromene derivatives with microtubule-destabilizing, anti-angiogenic, and MYB-inhibitory activities
20234 citationsauthor #7
Targeting Colon Cancer Cells with Pyrazino‐Imidazolinone Derivatives: Synthesis, Molecular Docking, and in Vitro Evaluation of Anti‐Proliferative and Pro‐Apoptotic Activities
20232 citationsauthor #7
New 4,5-Diarylimidazol-2-ylidene–iodidogold(I) Complexes with High Activity against Esophageal Adenocarcinoma Cells
20234 citationsauthor #9
Old Dogs with New Tricks: Antiparasitic Potential of Structurally Diverse 5-Nitrofuran and 5-Nitrothiophene Imines and Acyl Hydrazones
20231 citationsauthor #5
Editorial for the Special Issue—“Recent Advances of Novel Pharmaceutical Designs for Anti-Cancer Therapies”
20231 citationsauthor #1
Evaluation of the Antiparasitic and Antifungal Activities of Synthetic Piperlongumine‐Type Cinnamide Derivatives: Booster Effect by Halogen Substituents
202311 citationsauthor #14
Antitumor activity of the new tyrphostin briva against BRAFV600E-mutant colorectal carcinoma cells
20232 citationsauthor #7
A New Synthetic Curcuminoid Displays Antitumor Activities in Metastasized Melanoma
20239 citationsauthor #7
Fluorinated and N-Acryloyl-Modified 3,5-Di[(E)-benzylidene]piperidin-4-one Curcuminoids for the Treatment of Pancreatic Carcinoma
20237 citationsauthor #5
Versatile anti-infective properties of pyrido- and dihydropyrido[2,3-d]pyrimidine-based compounds.
20233 citationsauthor #11
Acryl-3,5-bis(2,4-difluorobenzylidene)-4-piperidone targeting cellular JUN proto-oncogene, AP-1 transcription factor subunit inhibits head and neck squamous cell carcinoma progression
20232 citationsauthor #9
Antitumor Effects of a New Retinoate of the Fungal Cytotoxin Illudin M in Brain Tumor Models
20224 citationsauthor #11
Novel Thienyl-Based Tyrosine Kinase Inhibitors for the Treatment of Hepatocellular Carcinoma
20224 citationsauthor #2
3D cell cultures, as a surrogate for animal models, enhance the diagnostic value of preclinical in vitro investigations by adding information on the tumour microenvironment: a comparative study of new dual-mode HDAC inhibitors
202211 citationsauthor #2
New chimeric HDAC inhibitors for the treatment of colorectal cancer
20228 citationsauthor #3
Antiparasitic activities of bimetallic N‐heterocyclic carbene gold(I) complexes with ferrocene ligands: relevance of chlorido and phosphino ligands
20221 citationsauthor #6
Targeting growth of breast cancer cell line (MCF-7) with curcumin-pyrimidine analogs
20224 citationsauthor #5
Immunomodulatory properties of HDAC6 inhibitors in cancer diseases: New chances for sophisticated drug design and treatment optimization.
202218 citationsauthor #1
2‐Amino‐4‐aryl‐5‐oxo‐4,5‐dihydropyrano[3,2‐c]chromene‐3‐carbonitriles with Microtubule‐Disruptive, Centrosome‐Declustering, and Antiangiogenic Effects in vitro and in vivo
20223 citationsauthor #5
Highly Efficient Single A3-Coupling (Aldehyde-Amine-Alkyne) Reaction Catalyzed by Air Stable Silver-(N-Heterocyclic Carbene) Complexes: Synthesis and Characterization
20221 citationsauthor #6
Doublecortin‐like kinase 1 is a therapeutic target in squamous cell carcinoma
20229 citationsauthor #24
Activity of Benzimidazole Derivatives and their N-Heterocyclic Carbene Silver Complexes Against Leishmania major Promastigotes and Amastigotes
20226 citationsauthor #8
A New Naphthopyran Derivative Combines c-Myb Inhibition, Microtubule-Targeting Effects, and Antiangiogenic Properties.
20227 citationsauthor #9
Chimeric HDAC and the cytoskeleton inhibitor broxbam as a novel therapeutic strategy for liver cancer
20224 citationsauthor #8
End Group Dye-labeled Polycarbonate Block Copolymers for Micellar (immuno-)Drug Delivery.
202216 citationsauthor #12
HDAC inhibitors with potential to overcome drug resistance in castration-resistant prostate cancer
202231 citationsauthor #1
Garcinol from Garcinia indica inhibits HIV‐1 reverse transcriptase‐associated ribonuclease H
20219 citationsauthor #6
p-Trifluoromethyl- and p-pentafluorothio-substituted curcuminoids of the 2,6-di[(E)-benzylidene)]cycloalkanone type: Syntheses and activities against Leishmania major and Toxoplasma gondii parasites.
202116 citationsauthor #13
A New Pentafluorothio-Substituted Curcuminoid with Superior Antitumor Activity
202113 citationsauthor #9
Activity of Fluorinated Curcuminoids against Leishmania major and Toxoplasma gondii Parasites
20213 citationsauthor #5
DNA as a Natural Flame Retardant for Cellulose Acetate Polymer Mixtures
202111 citationsauthor #10
Imidazole Analogs of Vascular-Disrupting Combretastatin A-4 with Pleiotropic Efficacy against Resistant Colorectal Cancer Models
20217 citationsauthor #2
Improved Anticancer Activities of a New Pentafluorothio-Substituted Vorinostat-Type Histone Deacetylase Inhibitor
20217 citationsauthor #9
Condensation of Lactones with Primary Diamines
20213 citationsauthor #5
Bcr-TMP, a Novel Nanomolar-Active Compound That Exhibits Both MYB- and Microtubule-Inhibitory Activity
202113 citationsauthor #9
An Update on Natural Antileishmanial Treatment Options from Plants, Fungi and Algae
202123 citationsauthor #5
New 3-Aryl-2-(2-thienyl)acrylonitriles with High Activity Against Hepatoma Cells
202110 citationsauthor #11
Anticancer Activity and Mechanisms of Action of New Chimeric EGFR/HDAC-Inhibitors
202120 citationsauthor #2
Front Cover: Activity of Fluorinated Curcuminoids against Leishmania major and Toxoplasma gondii Parasites (Chem. Biodiversity 9/2021)
20210 citationsauthor #5
3,3’-Diindolylmethane and its derivatives: nature-inspired strategies tackling drug resistant tumors by regulation of signal transduction, transcription factors and microRNAs
202019 citationsauthor #1
Evaluation of the antiparasitic activities of imidazol‐2‐ylidene–gold(I) complexes
202017 citationsauthor #8
Anticancer Active Heterocyclic Chalcones: Recent Developments.
202023 citationsauthor #5
Anticancer properties of chimeric HDAC and kinase inhibitors.
202048 citationsauthor #1
Guided Antitumoural Drugs: (Imidazol‐2‐ylidene)(L)gold(I) Complexes Seeking Cellular Targets Controlled by the Nature of Ligand L
20208 citationsauthor #8
New Pyrano‐4H‐benzo[g]chromene‐5,10‐diones with Antiparasitic and Antioxidant Activities
202014 citationsauthor #10
Investigation of melamine and DOPO-derived flame retardants for the bioplastic cellulose acetate
202014 citationsauthor #8
Synthesis and bioevaluation of new vascular-targeting and anti-angiogenic thieno[2,3-d]pyrimidin-4(3H)-ones.
202013 citationsauthor #7
Chemical and Biological Aspects of Garcinol and Isogarcinol: Recent Developments
201954 citationsauthor #2
A new 4-(pyridinyl)-4H-benzo[g]chromene-5,10-dione ruthenium(II) complex inducing senescence in 518A2 melanoma cells
201912 citationsauthor #7
New pyranoquinoline derivatives as vascular-disrupting anticancer agents
201911 citationsauthor #3
Antiparasitic activities of new lawsone Mannich bases
201926 citationsauthor #9
Alkylating anticancer agents and their relations to microRNAs
20198 citationsauthor #1
New naphthopyran analogues of LY290181 as potential tumor vascular-disrupting agents.
201927 citationsauthor #5
Garcinol Sensitizes NSCLC Cells to Standard Therapies by Regulating EMT-Modulating miRNAs
201948 citationsauthor #7
Pentafluorophenyl Substitution of Natural Di(indol‐3‐yl)methane Strongly Enhances Growth Inhibition and Apoptosis Induction in Various Cancer Cell Lines
20199 citationsauthor #7
New Antiparasitic Bis‐Naphthoquinone Derivatives
201919 citationsauthor #7
Discovery of natural products with metal-binding properties as promising antibacterial agents
201921 citationsauthor #4
Differential Methylation and Acetylation as the Epigenetic Basis of Resveratrol’s Anticancer Activity
201948 citationsauthor #6
Oxazole-Bridged Combretastatin A-4 Derivatives with Tethered Hydroxamic Acids: Structure–Activity Relations of New Inhibitors of HDAC and/or Tubulin Function
201925 citationsauthor #7
Anticancer properties of a new non-oxido vanadium(IV) complex with a catechol-modified 3,3'-diindolylmethane ligand.
201929 citationsauthor #4
Current State of Platinum Complexes for the Treatment of Advanced and Drug-Resistant Breast Cancers.
20197 citationsauthor #1
Antitumor and antiangiogenic activity of the novel chimeric inhibitor animacroxam in testicular germ cell cancer
201922 citationsauthor #6
Halogenated Bis(methoxybenzylidene)‐4‐piperidone Curcuminoids with Improved Anticancer Activity
201812 citationsauthor #7
Interplay of non-coding RNAs and approved antimetabolites such as gemcitabine and pemetrexed in mesothelioma
20185 citationsauthor #1
New (arene)ruthenium(II) complexes of 4‑aryl‑4H‑naphthopyrans with anticancer and anti-vascular activities.
201819 citationsauthor #6
Relations between approved platinum drugs and non-coding RNAs in mesothelioma
201813 citationsauthor #1
Recent developments concerning the application of the Mannich reaction for drug design
201843 citationsauthor #1

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