1,3,4-oxadiazole: a privileged structure in antiviral agents.

No abstract is available for this paper.

• Publication year

  2011

• Venue

  Mini-Reviews in Medical Chemistry

• Publication date

  2011-10-31

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.2174/138955711797655407PMID 22353222
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Functional roles of azoles motif in anti-HIV agents.

  2011cited by this paper
• Cosalane and its analogues: a unique class of anti-HIV agents.

  2010cited by this paper
• Crystal structures of HIV-1 reverse transcriptase with etravirine (TMC125) and rilpivirine (TMC278): implications for drug design.

  2010cited by this paper
• 1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 position.

  2009cited by this paper
• Efficient drug lead discovery and optimization.

  2009cited by this paper
• The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore.

  2009cited by this paper
• Raltegravir, elvitegravir, and metoogravir: the birth of "me-too" HIV-1 integrase inhibitors

  2009cited by this paper
• Crystallographic study of a novel subnanomolar inhibitor provides insight on the binding interactions of alkenyldiarylmethanes with human immunodeficiency virus-1 reverse transcriptase.

  2009influential reference
• Novel macrocyclic inhibitors of hepatitis C NS3/4A protease featuring a 2-amino-1,3-thiazole as a P4 carbamate replacement.

  2009influential reference
• Molecular modeling based approach to potent P2-P4 macrocyclic inhibitors of hepatitis C NS3/4A protease.

  2008cited by this paper
• Mutations in Human Immunodeficiency Virus Type 1 Integrase Confer Resistance to the Naphthyridine L-870,810 and Cross-Resistance to the Clinical Trial Drug GS-9137

  2008cited by this paper
• Efficient One-Pot Synthesis of Substituted 2-Amino-1,3,4-oxadiazoles.

  2008cited by this paper
• Synthesis and antiviral activity of azoles obtained from carbohydrates.

  2008cited by this paper
• Optimization of azoles as anti-human immunodeficiency virus agents guided by free-energy calculations.

  2008cited by this paper
• One-pot synthesis, antibacterial and antifungal activities of novel 2,5-disubstituted- 1,3,4-oxadiazoles

  2008cited by this paper
• Synthesis and Antiviral Evaluation of Novel 5‐(N‐Aryl‐aminomethyl‐1,3,4‐oxadiazol‐2‐yl)hydrazines and Their Sugars, 1,2,4‐Triazoles, Tetrazoles and Pyrazolyl Derivatives

  2008cited by this paper
• A new series of 2,5-bis(4-methylphenyl)-1,3,4-oxadiazole derivatives: their synthesis and fluorescence properties for anion sensors

  2007cited by this paper
• Synthesis and biological evaluation of alkenyldiarylmethane HIV-1 non-nucleoside reverse transcriptase inhibitors that possess increased hydrolytic stability.

  2007cited by this paper
• From docking false-positive to active anti-HIV agent.

  2007cited by this paper
• Privileged structures: a useful concept for the rational design of new lead drug candidates.

  2007cited by this paper
• Synthesis and properties of 1,3,4-oxadiazole-containing high-performance bismaleimide resins

  2007cited by this paper
• Molecular wires comprising pi-extended ethynyl- and butadiynyl-2,5-diphenyl-1,3,4-oxadiazole derivatives: synthesis, redox, structural, and optoelectronic properties.

  2006cited by this paper
• Synthesis and the biological evaluation of 2-benzenesulfonylalkyl-5-substituted-sulfanyl-[1,3,4]-oxadiazoles as potential anti-hepatitis B virus agents.

  2006cited by this paper
• Solid-phase synthesis of 1,3,4-oxadiazoline-5-thione derivatives from resin-bound acylhydrazines.

  2006cited by this paper
• Antiviral prodrugs – the development of successful prodrug strategies for antiviral chemotherapy

  2006cited by this paper
• One pot direct synthesis of oxazolines, benzoxazoles, and oxadiazoles from carboxylic acids using the Deoxo-Fluor reagent

  2006cited by this paper
• 1,3,4-Oxadiazole formation as traceless release in solid phase organic synthesis

  2006cited by this paper
• A simple and efficient one step synthesis of 1,3,4-oxadiazoles utilizing polymer-supported reagents and microwave heating

  2006cited by this paper
• Synthesis, Antimicrobial and Anti‐HIV Activity of Some Novel Benzenesulfonamides Bearing 2,5‐Disubstituted‐1,3,4‐Oxadiazole Moiety

  2006cited by this paper
• A mild and efficient one pot synthesis of 1,3,4-oxadiazoles from carboxylic acids and acyl hydrazides

  2006cited by this paper
• Novel HIV-1 integrase inhibitors derived from quinolone antibiotics.

  2006cited by this paper
• Synthesis, anti-HIV activity, and metabolic stability of new alkenyldiarylmethane HIV-1 non-nucleoside reverse transcriptase inhibitors.

  2005cited by this paper
• Synthesis of some new biologically active 1,3,4-oxadiazolyl nitroindoles and a modified Fischer indole synthesis of ethyl nitro indole-2-carboxylates.

  2005cited by this paper
• P1' oxadiazole protease inhibitors with excellent activity against native and protease inhibitor-resistant HIV-1.

  2004influential reference
• Synthesis, antimicrobial, and anti-HIV-1 activity of certain 5-(1-adamantyl)-2-substituted thio-1,3,4-oxadiazoles and 5-(1-adamantyl)-3-substituted aminomethyl-1,3,4-oxadiazoline-2-thiones.

  2004cited by this paper
• Synthesis, Characterization and Biological Activities of Substituted Oxadiazole, Triazole, Thiadiazole and 4‐Thiazolidinone Derivatives.

  2004cited by this paper
• Design, synthesis, anti-HIV activities, and metabolic stabilities of alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors.

  2004cited by this paper
• Dihydropyridine neuropeptide Y Y1 receptor antagonists 2. bioisosteric urea replacements.

  2004cited by this paper
• Efficient one-pot preparation of 5-substituted-2-amino-1,3,4-oxadiazoles using resin-bound reagents

  2004cited by this paper
• HIV-1 protease inhibitors with picomolar potency against PI-resistant HIV-1 by modification of the P1' substituent.

  2003cited by this paper
• The design, synthesis and evaluation of novel HIV-1 protease inhibitors with high potency against PI-resistant viral strains.

  2003cited by this paper
• Syntheses and insecticidal activity of new 2-(5-(trifluoromethyl)pyridyloxymethyl)-1,3,4-oxadiazoles

  2002cited by this paper
• New developments in anti-HIV chemotherapy.

  2002cited by this paper
• Newer N-substituted anthranilic acid derivatives as potent anti-inflammatory agents.

  2002cited by this paper
• New developments in anti-HIV chemotherapy

  2001cited by this paper
• AN EFFICIENT ONE POT SYNTHESIS OF 1,3,4-OXADIAZOLES

  2001cited by this paper
• New developments in anti-HIV chemotherapy

  2001cited by this paper
• A Mild Method for the Preparation of 1,3,4-Oxadiazoles: Triflic Anhydride Promoted Cyclization of Diacylhydrazines

  2000cited by this paper
• Syntheses and insecticidal activities of novel 2-fluorophenyl-5-aryl/cyclopropyl-1,3,4-oxadiazoles

  2000cited by this paper
• Trichloroacetic acid hydrazones I: New formation of 1,3,4-oxadiazoles from aldehydes

  1998cited by this paper
• Design, synthesis and antiinflammatory activity of some 1,3,4-oxadiazole derivatives.

  1997cited by this paper
• SYNTHESIS OF 2,5-DISUBSTITUTED-1,3,4-OXADIAZOLE, 1,5-DISUBSTITUTED-2-MERCAPTO-1,3,4-TRIAZOLE AND 2,5-DISUBSTITUTED-1,3,4-THIADIAZOLE DERIVATIVES AS PO TENTIAL ANTIMICROBIAL AGENTS

  1996cited by this paper
• Synthesis of 2,5‐Disubstituted‐1,3,4‐oxadiazole, 1,5‐Disubstituted‐2‐ mercapto‐1,3,4‐triazole and 2,5‐Disubstituted‐1,3,4‐thiadiazole Derivatives as Potential Antimicrobial Agents.

  1996cited by this paper
• The PETT series, a new class of potent nonnucleoside inhibitors of human immunodeficiency virus type 1 reverse transcriptase

  1995cited by this paper
• Synthesis and Antiinflammatory Activity of Some 3-Heterocyclyl-1,2- benzisothiazoles.

  1994cited by this paper
• Synthesis of unsymmetrically substituted 4 H -1,2,4-triazoles

  1994cited by this paper
• Synthesis and Antiinflammatory Activity of Some 3‐Heterocyclic Substituted 1,2‐Benzisothiazoles and 1,2,4‐Triazolo(4,3‐b)(1,2) benzisothiazoles.

  1992cited by this paper
• 2-(oxadiazolyl)- and 2-(thiazolyl)imidazo[1,2-a]pyrimidines as agonists and inverse agonists at benzodiazepine receptors.

  1991cited by this paper
• Synthesis and spectral data of 4,5-bis[5-aryl-1,3,4-oxadiazol-2-yl]-1-benzyl-1,2,3-triazoles

  1990cited by this paper
• A Convenient Synthesis of Alkyl and Aryl Substituted Bis-1,3,4-oxadiazoles

  1990cited by this paper
• SYNTHESIS OF SUBSTITUTED OXADIAZOLES, THIADIAZOLES AND TRIAZOLES AND EVALUATION OF THEIR BIOLOGICAL ACTIVITY

  1984cited by this paper
• Synthesis of 5-aryl-2-oxazolepropionic acids and analogs. Antiinflammatory agents

  1969cited by this paper
• Synthesis of 2,5-Bis(polyfluoroalkyl)-1,3,4-oxadiazoles and -thiadiazoles

  1961cited by this paper
• Zur acylierung von 5-aryl-tetrazolen; ein duplikationsverfahren zur darstellung von polyarylen☆

  1960cited by this paper
• Quaternary Salt Formation of Substituted Oxazoles and Thiazoles1

  1960cited by this paper
• Synthesis of Carboxylic Acid Hydrazides and s-Triazoles of the Anthraquinone Series

  1958cited by this paper
• 2,5-DIARYLOXAZOLES AND 2,5-DIARYL-1,3,4-OXADIAZOLES

  1955cited by this paper

• Quinoline-2-carboxlic acid derivatives bearing oxadiazole moiety: Synthesis, Skin Antitumor, ‎Antibacterial, antifungal activities, and POM studies for the Identification of the Pharmacophore ‎Sites

  2025cites this paper
• Synthesis, in vitro and in silico anticancer evaluations of novel styryl 1,3,4-oxadiazole-sulfonamide hybrids for colorectal cancer.

  2025cites this paper
• Synthesis, Antimicrobial Activity and Molecular Docking of New N-Acylated Derivatives of 5-(3-Phenoxyphenyl)-1,3,4-oxadiazol-2-amine

  2025cites this paper
• Development in medicinal chemistry via oxadiazole derivatives: patent spotlight 2020-2024.

  2025cites this paper
• Exploration of novel isoniazid embedded 1,3,4-oxadiazole hybrids as anti-TB, antioxidant, and COX inhibitors: synthesis, spectral analysis, and molecular modeling studies

  2025cites this paper
• Pd-, Cu-, and Ni-Catalyzed Reactions: A Comprehensive Review of the Efficient Approaches towards the Synthesis of Antibacterial Molecules

  2024cites this paper
• Design, Synthesis of Flurbiprofen Based 1,3,4‐Oxadiazoles and Constrained Anticancer, Antioxidant Agents: In silico Docking Analysis

  2024cites this paper
• UNVEILING THE POTENTIAL OF OXADIAZOLE TRIAZINE NUCLEOSIDE DERIVATIVE AS AN INHIBITOR OF SARS COV-2: A COMPUTATIONAL BREAKTHROUGH

  2024cites this paper
• Substituent effects on Axial Chiral Compound Enantiomers: Synthesis and Crystal Structures of Axially Chiral 1,3,4-Oxadiazole Thioethers (Sulfones) based on 2,2′-Bipyridine

  2024cites this paper
• I2-Mediated Synthesis of 1,3,4-Oxa/thiadiazoles from Aroylhydrazide and Acetonitrile/Thioacetamide.

  2024cites this paper
• Ascorbic Acid: An Efficient Organocatalyst for the Synthesis of 2‐Amino‐1,3,4‐oxadiazoles and Thiadiazoles via C−X Bond Formation

  2024cites this paper
• Investigation of Novel 2‐(Chloromethyl)‐5‐(3, 5‐Disubstituted‐1H‐Indol‐2‐yl)‐1,3,4‐Oxadiazole Derivatives as In Vitro, and In Silico Bioactivity Potential: Anti‐inflammatory, Anti‐TB and Antioxidant Activities Study

  2024cites this paper
• Synthesis of Novel 2-Mercapto-1,3,4-Oxadiazole Derivatives as Potent Urease Inhibitors: In Vitro and In Silico Investigations

  2024cites this paper
• 1,3,4-Oxadiazole Scaffold in Antidiabetic Drug Discovery: An Overview.

  2024cites this paper
• Benzohydrazide as a good precursor for the synthesis of novel bioactive and anti-oxidant 2-phenyl-1,3,4-oxadiazol-aminoacid derivatives: Structural determination, biological and anti-oxidant activity

  2024cites this paper
• Synthetic marvels in tuberculosis research: An in-depth review of 1,3,4-oxadiazole derivatives as antitubercular agents

  2024cites this paper
• Investigations of p-tolyloxy-1,3,4-oxadiazole propionamides as soybean 15-lipoxygenase inhibitors in comforting with in vitro and in silico studies

  2023cites this paper
• Mn(II) assisted synthesis of N-phenyl-5-(pyridin-3-yl)-1,3,4-oxadiazol-2-amine and evaluation of its Antiproliferative activity

  2023cites this paper
• Synthesis of Some New 1,3,4-Thiadiazole Derivatives Derived from Cholic Acid and Evaluation of their Biological Activity

  2023cites this paper
• Electrochemical Synthesis of N-Substituted 5-(1H-Indol-3-yl)-1,3,4-oxadiazole-2-amines: A Mild and Green Approach

  2023cites this paper
• A Comprehensive Review on the Antidiabetic Activity of Oxadiazole Derivatives

  2023cites this paper
• Crystal structure of 2-[(4-bromobenzyl)thio]-5-(5-bromothiophen-2-yl)-1,3,4-oxadiazole, C13H8Br2N2OS2

  2023cites this paper
• Protective effect of symmetrical N‐heterocyclic 1,3,4‐oxadiazole and 1,3,4‐thiadiazole derivatives against Pepino mosaic virus of tomato

  2022cites this paper
• Synthesis of Novel 1,3,4-Oxadiazole-Derived α-Aminophosphonates/α-Aminophosphonic Acids and Evaluation of Their In Vitro Antiviral Activity against the Avian Coronavirus Infectious Bronchitis Virus

  2022cites this paper
• Recent Advancement in Synthesis and Bioactivities of 1,3,4-Oxadiazole.

  2022cites this paper
• Cytotoxic Activity and Docking Studies of 2-arenoxybenzaldehyde N-acyl Hydrazone and 1,3,4-Oxadiazole Derivatives against Various Cancer Cell Lines

  2022cites this paper
• Synthesis, characterization, anti-mycobacterial activity and in silico study of new 2,5-disubstituted-1,3,4-oxadiazole derivatives.

  2022cites this paper
• A One-Pot Synthesis-Functionalization Strategy for Streamlined Access to 2,5-Disubstituted 1,3,4-Oxadiazoles from Carboxylic Acids

  2022cites this paper
• L-proline catalyzed ring transformation of 5-substituted tetrazole to 1,3,4-oxadiazoles as anti-tubercular agents

  2022cites this paper
• 1,3,4‐oxadiazole derivatives as potential antimicrobial agents

  2022cites this paper
• Potential Synthetic Routes and Metal-Ion Sensing Applications of 1,3,4-Oxadiazoles: An Integrative Review

  2022cites this paper
• Oxadiazole derivatives: Histone Deacetylase Inhibitors in anticancer therapy and drug discovery

  2022cites this paper
• Flow synthesis of oxadiazoles coupled with sequential in-line extraction and chromatography

  2022cites this paper
• Review of the biological activities of heterocyclic compounds comprising oxadiazole moieties.

  2022cites this paper
• Pyrimidine-fused Dinitrogenous Penta-heterocycles as a Privileged Scaffold for Anti-Cancer Drug Discovery.

  2022cites this paper
• Synthesis of 7-Azaindole Based Carbohydrazides and 1,3,4-Oxadiazoles; Antioxidant Activity, α-Glucosidase Inhibition Properties and Docking Study

  2022cites this paper
• Oxadiazoles for Covid-19?

  2021cites this paper
• Synthesis, spectroscopic characterization and DNA/HSA binding studies of (phenyl/naphthyl)ethenyl-substituted 1,3,4-oxadiazolyl-1,2,4-oxadiazoles

  2021cites this paper
• In Vitro and In Silico Evaluation of Biological Properties of Some 1, 3, 4-Oxadiazole Derivatives Against Streptococcus mutans and Their Interaction With Gbp-C by Molecular Docking

  2021cites this paper
• Synthetic Coumarin Derivatives as SARS‐CoV‐2 Major Protease Inhibitors: Design, Synthesis, Bioevaluation and Molecular Docking

  2021cites this paper
• SET activation of nitroarenes by 2-azaallyl anions as a straightforward access to 2,5-dihydro-1,2,4-oxadiazoles

  2021cites this paper
• The Fellowship of Privileged Scaffolds—One Structure to Inhibit Them All

  2021cites this paper
• A novel dipeptide coupled with pyrazine-oxadiazole derivative as a potential antitubercular agent: Synthesis, radioiodination and bioevaluation.

  2021cites this paper
• Synthesis of pyrrolo[3,2-c]carbazole-2-carbohydrazides and pyrrolo[3,2-c]carbazol-2-yl-1,3,4-oxadiazoles and their in vitro antibacterial evaluation

  2021cites this paper
• A Three-Component Ugi-Type Reaction of N-Carbamoyl Imines Enables a Broad Scope Primary α-Amino 1,3,4-Oxadiazole Synthesis.

  2021cites this paper
• Design, synthesis, modelling studies and biological evaluation of 1,3,4-oxadiazole derivatives as potent anticancer agents targeting thymidine phosphorylase enzyme.

  2021cites this paper
• Visible-Light Photocatalytic Ugi/Aza-Wittig Cascade towards 2-Aminomethyl-1,3,4-oxadiazole Derivatives

  2021cites this paper
• Efficient Synthesis of Novel N-[4-Methyl-3-(4-(5-phenyl-1,3,4-oxadiazol-2-yl)phenyl)thiazol-2(3H)-ylidene]benzamide Hybrid Ring System as Potential Antibacterial Agents.

  2021cites this paper
• Synthesis of trans- methyl ferulate bearing an oxadiazole ether as potential activators for controlling plant virus.

  2021cites this paper
• General α‐Amino 1,3,4‐Oxadiazole Synthesis via Late‐Stage Reductive Functionalization of Tertiary Amides and Lactams

  2021cites this paper
• Electrosynthesis of 2-(1,3,4-Oxadiazol-2-yl)aniline Derivatives with Isatins as Amino-attached C1 Sources.

  2020cites this paper
• Design, Synthesis and Pharmacological evalution of 1,3,4-Oxadiazole Derivatives As Collapsin Response Mediator Protein 1 (CRMP 1) Inhibitors.

  2020cites this paper
• Novel Bi-heterocycles as Potent Inhibitors of Urease and Less Cytotoxic Agents: 3-({5-((2-Amino-1,3-thiazol-4-yl)methyl)-1,3,4-oxadiazol-2-yl}sulfanyl)-N-(un/substituted-phenyl)propanamides

  2020cites this paper
• SYNTHESIS AND ANTI-PROLIFERATIVE SCREENING OF NEW THIAZOLE COMPOUNDS

  2020cites this paper
• Synthesis of Novel Bi-Heterocycles as Valuable Anti-Diabetic Agents: 2-({5-((2-Amino-1,3-Thiazol-4-yl)methyl)-1,3,4-Oxadiazol-2-yl}sulfanyl)-N-(Substituted)acetamides

  2020cites this paper
• Determination of potential inhibitors based on isatin derivatives against SARS-CoV-2 main protease (mpro): a molecular docking, molecular dynamics and structure-activity relationship studies

  2020influential citation
• Structure-based drug designing of naphthalene based SARS-CoV PLpro inhibitors for the treatment of COVID-19

  2020cites this paper
• Synthesis, telomerase inhibitory and anticancer activity of new 2-phenyl-4H-chromone derivatives containing 1,3,4-oxadiazole moiety

  2020cites this paper
• CHLORAMINE-T MEDIATED SYNTHESIS OF 1,3,4-OXADIAZOLE DERIVATIVES

  2020cites this paper
• Design, Synthesis, Antimicrobial Evaluation, and Laccase Catalysis Effect of Novel Benzofuran–Oxadiazole and Benzofuran–Triazole Hybrids

  2019cites this paper
• 1,3,4-Oxadiazoles by Ugi-Tetrazole and Huisgen Reaction

  2019cites this paper
• Spectroscopic, DFT studies and electronic properties of novel functionalized bis-1,3,4-thiadiazoles

  2019cites this paper
• [3 + 2]-Cycloaddition of 2 H-Azirines with Nitrosoarenes: Visible-Light-Promoted Synthesis of 2,5-Dihydro-1,2,4-oxadiazoles.

  2019cites this paper
• Design, synthesis, antimicrobial evaluation, and molecular docking studies of novel symmetrical 2,5‐difunctionalized 1,3,4‐oxadiazoles

  2019cites this paper
• Sequential Multicomponent Synthesis of 2-(Imidazo[1,5-α]pyridin-1-yl)-1,3,4-Oxadiazoles

  2019cites this paper
• A transition metal-free approach towards synthesis of β-carboline tethered 1,3,4-oxadiazoles via oxidative C–O bond formation

  2019cites this paper
• Overview of Recent Strategic Advances in Medicinal Chemistry.

  2019cites this paper
• Synthesis of N-pyrimidin[1,3,4]oxadiazoles and N-pyrimidin[1,3,4]-thiadiazoles from 1,3,4-oxadiazol-2-amines and 1,3,4-thiadiazol-2-amines via Pd-catalyzed heteroarylamination

  2019cites this paper
• Design, synthesis, neuroprotective, antibacterial activities and docking studies of novel thieno[2,3-d]pyrimidine-alkyne Mannich base and oxadiazole hybrids.

  2018cites this paper
• N-[2-(1H-Indol-3-yl)-1-(5-thioxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)ethyl]-4-methylbenzenesulfonamide

  2018cites this paper
• Current insights into anti-HIV drug discovery and development: a review of recent patent literature (2014–2017)

  2018cites this paper
• 2-(5-Methyl-1-phenyl-1H-1,2,3-triazol-4-yl)-5-phenyl-1,3,4-oxadiazole

  2018cites this paper
• Synthesis, biological evaluation, and molecular docking study of pyridine clubbed 1,3,4-oxadiazoles as potential antituberculars

  2018cites this paper
• Synthesis and Anti-H5N1 Activity of Substituted Pyridine Glycosides and (Oxadiazolyl)oxymethylpyridine Acyclic C-Nucleoside Analogues

  2018cites this paper
• Synthesis, in vitro and in silico studies of novel potent urease inhibitors: N-[4-({5-[(3-Un/substituted-anilino-3-oxopropyl)sulfanyl]-1,3,4-oxadiazol-2-yl}methyl)-1,3-thiazol-2-yl]benzamides.

  2018cites this paper
• Current Parallel Solid-Phase Synthesis of Drug-like Oxadiazole and Thiadiazole Derivatives for Combinatorial Chemistry.

  2018cites this paper
• DESIGN AND SYNTHESIS OF NOVEL 1,3,4-OXADIAZOLE AND 1,2,4-TRIAZOLO[3,4- B]1,3,4-THIADIAZOLE DERIVATIVES AND THEIR ANTIMICROBIAL STUDIES

  2018cites this paper
• Antimicrobial evaluation and action mechanism of pyridinium-decorated 1,4-pentadien-3-one derivatives.

  2018cites this paper
• Design, synthesis and pharmacological studies of some new quinoline Schiff bases and 2,5-(disubstituted-[1,3,4])-oxadiazoles

  2017cites this paper
• Highly Efficient One-Pot Solvent-Free Synthesis of 2,5-Disubstituted-1,3,4-Oxadiazole via BTI-mediated Oxidation of N-Acylhydrazone from Hydrazide and Aldehyde

  2017cites this paper
• Design, synthesis and biological evaluation of imidazopyridine-propenone conjugates as potent tubulin inhibitors.

  2017cites this paper
• Benzisoxazole: a privileged scaffold for medicinal chemistry.

  2017cites this paper
• Synthesis of Oxadiazolyl, Pyrazolyl and Thiazolyl Derivatives of Thiophene-2-Carboxamide as Antimicrobial and Anti-HCV Agents

  2017cites this paper
• Identification of spirocyclic or phosphate substituted quinolizine derivatives as novel HIV-1 integrase inhibitors: a patent evaluation of WO2016094197A1, WO2016094198A1 and WO2016154527A1

  2017cites this paper
• Chalcone: A Privileged Structure in Medicinal Chemistry.

  2017cites this paper
• Synthesis of novel 1,3,4-oxadiazole derivatives containing diamides as promising antibacterial and antiviral agents

  2017cites this paper
• Antiviral and Antibacterial Activities of N‐(4‐Substituted phenyl) Acetamide Derivatives Bearing 1,3,4‐Oxadiazole Moiety

  2016cites this paper
• Synthesis and antioxidant evaluation of some new 2-benzoylamino-5-hetaryl-1,3,4-oxadiazoles

  2016cites this paper
• Synthesis and biological evaluation of imidazopyridinyl-1,3,4-oxadiazole conjugates as apoptosis inducers and topoisomerase IIα inhibitors.

  2016cites this paper
• Iodine-Mediated Domino Oxidative Cyclization: One-Pot Synthesis of 1,3,4-Oxadiazoles via Oxidative Cleavage of C(sp(2))-H or C(sp)-H Bond.

  2016cites this paper
• Synthesis and Antimicrobial Evaluation of Symmetrical Diquaternary Ammonium Salts Bearing Bis-1,3,4-Oxadiazole Rings Moieties

  2016cites this paper
• Intramolecular decarboxylative coupling as the key step in copper-catalyzed domino reaction: facile access to 2-(1,3,4-oxadiazol-2-yl)aniline derivatives.

  2015cites this paper
• Therapeutic efficacy of liposomes containing 4-(5-pentadecyl-1,3,4-oxadiazol-2-yl)pyridine in a murine model of progressive pulmonary tuberculosis.

  2015cites this paper
• Base as Potential Antimicrobial and Antiproliferative Agents

  2015cites this paper
• Synthesis and Anti‐cancer Activity of 1,3,4‐Thiadiazole and 1,3‐Thiazole Derivatives Having 1,3,4‐Oxadiazole Moiety

  2015cites this paper
• Synthesis and Anti‐Hepatitis B Virus Evaluation of 7‐Methoxy‐3‐heterocyclic quinolin‐6‐ols

  2015cites this paper
• Synthesis of 2-amino-1,3,4-oxadiazoles and 2-amino-1,3,4-thiadiazoles via sequential condensation and I2-mediated oxidative C–O/C–S bond formation.

  2015cites this paper
• Synthesis of Novel Trifluorobenzimidazole Derivatives and Their Study of 5-LOX Inhibition and Brine Shrimp Lethal Bioassay (BSLB)

  2015cites this paper
• Synthesis of Novel 2,5-Disubstituted-1,3,4-thiadiazoles Clubbed 1,2,4-Triazole, 1,3,4-Thiadiazole, 1,3,4-Oxadiazole and/or Schiff Base as Potential Antimicrobial and Antiproliferative Agents

  2015cites this paper
• Palladium-catalyzed one-pot synthesis of diazoles via tert-butyl isocyanide insertion.

  2015cites this paper