Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.

No abstract is available for this paper.

• Publication year

  2014

• Venue

  Journal of Medicinal Chemistry

• Publication date

  2014-07-07

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1021/jm5005489PMID 24918545
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Pharmacologic profiles of investigational kisspeptin/metastin analogues, TAK-448 and TAK-683, in adult male rats in comparison to the GnRH analogue leuprolide.

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