Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?

No abstract is available for this paper.

• Publication year

  1990

• Venue

  Journal of Medicinal Chemistry

• Publication date

  Unknown publication date

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1021/JM00163A001PMID 1967317
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

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• A highly potent and selective H3 agonist relaxes rabbit middle cerebral artery, in vitro.

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  1988cited by this paper
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• Inhibition of guinea pig ileum contractions mediated by a class of histamine receptor resembling the H3 subtype.

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• Stereoselectivity of the histamine H3-presynaptic autoreceptor.

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• Actions of betahistine at histamine receptors in the brain.

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• Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

  1983cited by this paper
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• Species-related pharmacological heterogeneity of histamine H(3) receptors.

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  1999cites this paper
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  1999cites this paper
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  1998cites this paper
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  1998cites this paper
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  1998cites this paper
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  1998cites this paper
• The intradermal effects of the H3 receptor agonist R α methylhistamine in human skin

  1998cites this paper
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  1998cites this paper
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  1998cites this paper
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  1998cites this paper
• High antagonist potency of GT-2227 and GT-2331, new histamine H3 receptor antagonists, in two functional models.

  1998cites this paper
• DNA-chlorpheniramine interaction studied by spectroscopic techniques.

  1998cites this paper
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