Scalable total syntheses of N-linked tryptamine dimers by direct indole-aniline coupling: psychotrimine and kapakahines B and F.

No abstract is available for this paper.

• Publication year

  2010

• Venue

  Journal of the American Chemical Society

• Publication date

  2010-05-26

• Fields of study

  Medicine, Chemistry

• Identifiers
  DOI 10.1021/ja1009458PMID 20426477PMCID PMC2874090
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar, PubMed

• No claims are published for this paper.

• No concepts are published for this paper.

• Stereocontrolled and efficient total synthesis of (-)-stephanotic acid methyl ester and (-)-celogentin C.

  2010cited by this paper
• On the absolute configurational stability of bromonium and chloronium ions.

  2010cited by this paper
• Total synthesis of kapakahine E and F.

  2010cited by this paper
• Total synthesis of the antimitotic bicyclic peptide celogentin C.

  2010cited by this paper
• Total synthesis of celogentin C by stereoselective C-H activation.

  2010cited by this paper
• Determination of absolute configuration of trimeric indole alkaloid, psychotrimine, by first asymmetric total synthesis.

  2010cited by this paper
• Catalytic oxyamidation of indoles.

  2010cited by this paper
• Enantiospecific total syntheses of kapakahines B and F.

  2009cited by this paper
• A straightforward total synthesis of (-)-chaetominine.

  2009cited by this paper
• Copper-mediated coupling of 1,1-dibromo-1-alkenes with nitrogen nucleophiles: a general method for the synthesis of ynamides.

  2009cited by this paper
• Total synthesis of (+)-haplophytine.

  2009cited by this paper
• Total Synthesis of (+)-11,11'-Dideoxyverticillin A

  2009cited by this paper
• Total synthesis of chloropeptin II (complestatin) and chloropeptin I.

  2009cited by this paper
• Observation of direct sulfenium and selenenium group transfer from thiiranium and seleniranium ions to alkenes.

  2009cited by this paper
• Total synthesis of vinblastine, vincristine, related natural products, and key structural analogues.

  2009cited by this paper
• Chemoselectivity: the mother of invention in total synthesis.

  2009cited by this paper
• Redox economy in organic synthesis.

  2009cited by this paper
• Total synthesis of (+)-haplophytine.

  2009cited by this paper
• Total synthesis of celogentin C.

  2009cited by this paper
• Protecting-group-free synthesis as an opportunity for invention.

  2009cited by this paper
• The mechanism of the oxidative polymerization of aniline and the formation of supramolecular polyaniline structures

  2008cited by this paper
• It all began with an error: the nomofungin/communesin story.

  2008cited by this paper
• Pyrrole-2-carboxylic acid as a ligand for the Cu-catalyzed reactions of primary anilines with aryl halides.

  2008cited by this paper
• Enantiospecific total synthesis of the hapalindoles, fischerindoles, and welwitindolinones via a redox economic approach.

  2008cited by this paper
• An expeditious synthesis of C(3)-N(1') heterodimeric indolines.

  2008cited by this paper
• Total synthesis of (+/-)-psychotrimine.

  2008cited by this paper
• Copper-catalyzed cyclization of iodo-tryptophans: a straightforward synthesis of pyrroloindoles.

  2008cited by this paper
• Facile and general synthesis of quaternary 3-aminooxindoles.

  2008cited by this paper
• Pestalazines and pestalamides, bioactive metabolites from the plant pathogenic fungus Pestalotiopsis theae.

  2008cited by this paper
• Mechanistic insights into the stereocontrolled synthesis of hexahydropyrrolo[2,3-b]indoles by electrophilic activation of tryptophan derivatives.

  2008cited by this paper
• Total synthesis of chaetominine.

  2008cited by this paper
• Stereoselective oxidative rearrangement of 2-aryl tryptamine derivatives.

  2008cited by this paper
• First total synthesis of trimeric indole alkaloid, psychotrimine.

  2008cited by this paper
• Synthesis of (-)-chaetominine.

  2007cited by this paper
• Total synthesis of marine natural products without using protecting groups

  2007cited by this paper
• Total synthesis of complex cyclotryptamine alkaloids: stereocontrolled construction of quaternary carbon stereocenters.

  2007cited by this paper
• Total synthesis of (+/-)-communesin F.

  2007cited by this paper
• Total synthesis of the opioid agonistic indole alkaloid mitragynine and the first total syntheses of 9-methoxygeissoschizol and 9-methoxy-Nb-methylgeissoschizol.

  2007cited by this paper
• Synthesis of indole alkaloid analogues containing the novel hexahydropyrrolo[1′,2′,3′:1,9a,9]imidazo[1,2-a]indole skeleton by ring-closing reactions of tryptophan-derived α-amino nitriles

  2007cited by this paper
• Chemistry of the Hexahydropyrrolo[2,3-b]indoles: configuration, conformation, reactivity, and applications in synthesis.

  2007cited by this paper
• Concise total synthesis of (-)-calycanthine, (+)-chimonanthine, and (+)-folicanthine.

  2007cited by this paper
• General approach for the synthesis of 12-methoxy-substituted sarpagine indole alkaloids including (-)-12-methoxy-N(b)-methylvoachalotine, (+)-12-methoxy-N(a)-methylvellosimine, (+)-12-methoxyaffinisine, and (-)-fuchsiaefoline.

  2006cited by this paper
• Chaetominine, a cytotoxic alkaloid produced by endophytic Chaetomium sp. IFB-E015.

  2006cited by this paper
• Bisindole alkaloids.

  2006cited by this paper
• Investigations of Pd-catalyzed ArX coupling reactions informed by reaction progress kinetic analysis.

  2006cited by this paper
• Total synthesis of (+/-)-chartelline C.

  2006cited by this paper
• Synthesis of the celogentin C right-hand ring.

  2006cited by this paper
• Synthesis and self-assembling properties of diacetylene-containing glycolipids.

  2006cited by this paper
• The structural and synthetic implications of the biosynthesis of the calycanthaceous alkaloids, the communesins, and nomofungin

  2006cited by this paper
• Chaetocochins A-C, epipolythiodioxopiperazines from Chaetomium cochliodes.

  2006cited by this paper
• Protecting-group-free synthesis

  2006cited by this paper
• High yielding synthesis of 3a-hydroxypyrrolo[2,3-b]indoline dipeptide methyl esters: synthons for expedient introduction of the hydroxypyrroloindoline moiety into larger peptide-based natural products and for the creation of tryptathionine bridges.

  2005cited by this paper
• A remarkable ring contraction en route to the chartelline alkaloids.

  2005cited by this paper
• Photogenerated N-methyl-N-1-naphthylnitrenium ion: laser flash photolysis, trapping rates, and product study.

  2005cited by this paper
• A general strategy for the synthesis of vincamajine-related indole alkaloids: stereocontrolled total synthesis of (+)-dehydrovoachalotine, (-)-vincamajinine, and (-)-11-methoxy-17-epivincamajine as well as the related quebrachidine diol, vincamajine diol, and vincarinol.

  2005cited by this paper
• Reaction progress kinetic analysis: a powerful methodology for mechanistic studies of complex catalytic reactions.

  2005cited by this paper
• m-chloroperbenzoic acid oxidation of corynanthe-type indole alkaloid, mitragynine, afforded unusual dimerization products

  2004cited by this paper
• New type of trimeric and pentameric indole alkaloids from Psychotria rostrata.

  2004cited by this paper
• Total synthesis of (+/-)-perophoramidine.

  2004cited by this paper
• Small molecule blockade of transcriptional coactivation of the hypoxia-inducible factor pathway.

  2004cited by this paper
• Regiospecific, enantiospecific total synthesis of the 12-alkoxy-substituted indole alkaloids, (+)-12-methoxy-Na-methylvellosimine, (+)-12-methoxyaffinisine, and (-)-fuchsiaefoline.

  2004cited by this paper
• Photodecomposition reaction of trapped aniline cation by photofragment excitation spectroscopy

  2004cited by this paper
• Synthesis of novel acetylene-containing amino acids

  2003cited by this paper
• Electronic structures, vibrational spectra, and revised assignment of aniline and its radical cation: Theoretical study

  2003cited by this paper
• Studies of the reactions between indole-2,3-diones (isatins) and 2-aminobenzylamine

  2003cited by this paper
• Chemoselectivity of the ruthenium-catalyzed hydrative diyne cyclization: total synthesis of (+)-cylindricine C, D, and E.

  2003cited by this paper
• More kapakahines from the marine sponge Cribrochalina olemda.

  2003cited by this paper
• Synthesis and antinociceptive activity of chimonanthines and pyrrolidinoindoline-type alkaloids.

  2002cited by this paper
• Reactions of N-methyl-N-(4-biphenylyl)nitrenium ion with electron-rich arenes: laser flash photolysis and product studies.

  2002cited by this paper
• The copper-catalyzed N-arylation of indoles.

  2002cited by this paper
• Recent Advances in the Chemistry of 1-Hydroxyindoles, 1-Hydroxytryptophans, and 1-Hydroxytryptamines

  2002cited by this paper
• Nucleophilic Substitution Reaction on the Nitrogen of Indole Nucleus: A Novel Synthesis of 1-Aryltryptamines

  2002cited by this paper
• Regiospecific, enantiospecific total synthesis of the alkoxy-substituted indole bases, 16-epi-N(a)-methylgardneral, 11-methoxyaffinisine, and 11-methoxymacroline as well as the indole alkaloids alstophylline and macralstonine.

  2002cited by this paper
• Dimerization of indole derivatives with hypervalent iodines(III): a new entry for the concise total synthesis of rac- and meso-chimonanthines

  2002cited by this paper
• Stereocontrolled total synthesis of (+)-vinblastine.

  2002cited by this paper
• Enantioselective total synthesis of quadrigemine C and psycholeine.

  2002cited by this paper
• Total synthesis of asperazine.

  2001cited by this paper
• Efficient asymmetric synthesis of biologically important tryptophan analogues via a palladium-mediated heteroannulation reaction.

  2001cited by this paper
• Discovery through total synthesis: a retrospective on the himastatin problem.

  2001cited by this paper
• An efficient synthesis of optically active physostigmine from tryptophan via alkylative cyclization.

  2000cited by this paper
• One-pot synthesis of unsymmetrical triarylamines from aniline precursors.

  2000cited by this paper
• Synthesis of Strychnine.

  2000cited by this paper
• Simple, efficient catalyst system for the palladium-catalyzed amination of aryl chlorides, bromides, and triflates.

  2000cited by this paper
• A convenient and scaleable procedure for removing the Fmoc group in solution

  2000cited by this paper
• On the Reaction of Tryptophan Derivatives with N-Phenylselenyl Phthalimide: The Nature of the Kinetic and Thermodynamic Hexahydropyrrolo[2,3-b]indole Products. Alkylation of Tryptophan with Inversion of Configuration

  1999cited by this paper
• Free-Radical Ring Contraction of Six-, Seven-, and Eight-Membered Lactones by a 1,2-Shift Mechanism. A Kinetic and (17)O NMR Spectroscopic Study.

  1999cited by this paper
• Total Synthesis of 5-N-Acetylardeemin and Amauromine: Practical Routes to Potential MDR Reversal Agents

  1999cited by this paper
• Chemical trapping experiments support a cation‐radical mechanism for the oxidative polymerization of aniline

  1999cited by this paper
• Synthesis of 5-, 6- and 7-azaindoles via palladium-catalyzed heteroannulation of internal alkynes

  1998cited by this paper
• Total Synthesis of Himastatin: Confirmation of the Revised Stereostructure.

  1998cited by this paper
• Synthesis of 2,3-Disubstituted Indoles via Palladium-Catalyzed Annulation of Internal Alkynes

  1998cited by this paper
• Studies in the Total Synthesis of Himastatin: A Revision of the Stereochemical Assignment.

  1998cited by this paper
• SUBSTITUENT EFFECTS ON THE LIFETIMES AND REACTIVITIES OF ARYLNITRENIUM IONS STUDIED BY LASER FLASH PHOTOLYSIS AND PHOTOTHERMAL BEAM DEFLECTION

  1996cited by this paper
• Stereocontrolled Total Syntheses of meso-Chimonanthine and meso-Calycanthine via a Novel Samarium Mediated Reductive Dialkylation

  1996cited by this paper
• The Kapakahines, Cyclic Peptides from the Marine Sponge Cribrochalina olemda.

  1996cited by this paper
• Acid−Base Properties of Arylnitrenium Ions

  1996cited by this paper
• Kapakahine B, a cyclic hexapeptide with an .alpha.-carboline ring system from the marine sponge Cribrochalina olemda

  1995cited by this paper
• A stereoselective transformation of pseudoindoxyls into oxindoles in a single operation

  1994cited by this paper
• Effect of tertiary bases on O-benzotriazolyluronium salt-induced peptide segment coupling

  1994cited by this paper
• Stereoselective Total Syntheses of Amauromine and 5-N-Acetylardeemin. A Concise Route to the Family of "Reverse-Prenylated" Hexahydropyrroloindole Alkaloids

  1994cited by this paper

• Trimeric natural products: structural diversity, biosynthesis, bioactivities and chemical synthesis.

  2026cites this paper
• Intra-/Intermolecular 1,2-Diamination of Alkenyl Oximes with O-Benzoylhydroxylamines Enabled by Copper Catalysis.

  2025cites this paper
• Sustainable Copper-Catalyzed Cyanation of Aryl Iodine through a Design of Experiment Strategy

  2025cites this paper
• Bioinspired Syntheses of the Marine Pyridoacridine Alkaloids 2-Bromo and 3-Bromodeoxyamphimedine and Structure Correction of 2-Bromoamphimedine.

  2025cites this paper
• Pd/BINAP/Peroxide‐Enabled Relay Multicomponent Reactions

  2025cites this paper
• Total Syntheses of Diketopiperazine Alkaloids via Divergent C3-N1' and C3-C5' Bond Anchor.

  2025cites this paper
• Atroposelective Total Synthesis of Cihunamide B.

  2024cites this paper
• Regioselective Brønsted acid catalyzed ring opening of aziridines by phenols and thiophenols; a gateway to access functionalized indolines, indoles, benzothiazines, dihydrobenzo-thiazines, benzo-oxazines and benzochromenes.

  2024cites this paper
• Modular, Scalable Total Synthesis of Lapparbin with a Noncanonical Biaryl Linkage.

  2024cites this paper
• Green Late-Stage Functionalization of Tryptamines.

  2024cites this paper
• Transition-Metal-Catalyzed 1,2-Diaminations of Olefins: Synthetic Methodologies and Mechanistic Studies.

  2023cites this paper
• Recent Advancements on Metal-Free Vicinal Diamination of Alkenes: Synthetic Strategies and Mechanistic Insights.

  2023cites this paper
• Mechanistic duality of indolyl 1,3-heteroatom transposition

  2023cites this paper
• Silver(I)/Dirhodium(II) Catalytic Platform for Asymmetric N-H Insertion Reaction of Heteroaromatics.

  2023cites this paper
• Dual Nickel/Photoredox‐Catalyzed Synthesis of N‐formyl N,N’‐Diaryl Ethylenediamines via Multiple C−N/C−C Coupling of Nitroarenes with Trimethylamine

  2023cites this paper
• Atroposelective Synthesis of Planar-Chiral Indoles via Carbene Catalyzed Macrocyclization.

  2023cites this paper
• POCl3/Sulfoxide-Promoted Synthesis of Indolizino[8,7-b]indoles.

  2023cites this paper
• Nitrite-catalyzed economic and sustainable bromocyclization of tryptamines/ tryptophols to access hexahydropyrrolo[2,3-b]indoles/tetrahydrofuroindolines in batch and flow

  2023cites this paper
• Sustainable Electrochemical Dearomatization for the Synthesis of Diverse 2,3-Functionalized Indolines

  2022cites this paper
• An N-N linked dimeric indole alkaloid from the marine sponge-associated rare actinomycetes Kocuria sp. S42

  2022cites this paper
• Copper-Mediated Single-Electron Approach to Indoline Amination: Scope, Mechanism, and Total Synthesis of Asperazine A.

  2022cites this paper
• Energy Transfer-Enabled Unsymmetrical Diamination Using Unprecedented Bifunctional Nitrogen-Radical Precursors

  2022cites this paper
• Energy transfer-enabled unsymmetrical diamination using bifunctional nitrogen-radical precursors

  2022cites this paper
• Total synthesis of (+)-asperazine A: A stereoselective domino dimerization

  2022cites this paper
• Atroposelective Total Synthesis of Darobactin A.

  2022cites this paper
• The tryptophan connection: cyclic peptide natural products linked via the tryptophan side chain.

  2021cites this paper
• Indole‐2‐Carboxaldehyde: An Emerging Precursor for the Construction of Diversified Imperative Skeleton

  2021cites this paper
• THE EFFICACY OF MARINE NATURAL PRODUCTS AGAINST PLASMODIUM FALCIPARUM.

  2021cites this paper
• Intramolecular Aminolactonization for Synthesis of Furoindolin-2-One

  2021cites this paper
• Catalytic Function of Cu (I) and Cu (II) in Total Synthesis of Alkaloids

  2021cites this paper
• Small-Scale Preparation of Fluorescently Labeled Chemical Probes from Marine Cyclic Peptides, Kapakahines A and F

  2021cites this paper
• Total Synthesis of Aetokthonotoxin, the Cyanobacterial Neurotoxin Causing Vacuolar Myelinopathy

  2021cites this paper
• Blue LED-Mediated N-H Insertion of Indoles into Aryldiazoesters at Room Temperature in Batch and Flow: Reaction Kinetics, Density Functional Theory, and Mechanistic Study.

  2021cites this paper
• Synthesis of Indoloquinolines: An Intramolecular Cyclization Leading to Advanced Perophoramidine-Relevant Intermediates

  2021cites this paper
• Synthesis and Activation of Bench-Stable 3a-Fluoropyrroloindolines as Latent Electrophiles for the Synthesis of C-2-Thiol-Substituted Tryptophans and C-3a-Substituted Pyrroloindolines.

  2019cites this paper
• Copper-catalyzed nitrene transfer/cyclization cascade to synthesize 3a-nitrogenous furoindolines and pyrroloindolines

  2019cites this paper
• Regiodivergent Intramolecular Nucleophilic Addition of Ketimines for the Diverse Synthesis of Azacycles.

  2019cites this paper
• Cytotoxic and antimicrobial indole alkaloids from an endophytic fungus Chaetomium sp. SYP-F7950 of Panax notoginseng

  2019cites this paper
• Controlling the regioselectivity of the ring opening of spiro-epoxyoxindoles for efficient synthesis of C(3)-N(1')-bisindoles and C(3)-N(1')-diindolylmethane.

  2019cites this paper
• Heteroaryl Rings in Peptide Macrocycles.

  2019cites this paper
• Rapid Generation of Molecular Complexity by Chemical Synthesis: Highly Efficient Total Synthesis of Hexacyclic Alkaloid (-)-Chaetominine and Its Biosynthetic Implications.

  2018cites this paper
• Enantioselective Bromocyclization of Tryptamines Induced by Chiral Co(III)-Complex-Templated Brønsted Acids under an Air Atmosphere.

  2018cites this paper
• Asymmetric Total Synthesis and Absolute Configuration Determination of (-)-Verrupyrroloindoline.

  2018cites this paper
• Photosensitized Cross-Linking of Tryptophan and Tyrosine Derivatives by Rose Bengal in Aqueous Solutions.

  2018cites this paper
• Lipase-catalyzed kinetic resolution approach toward enantiomerically enriched 1-(β-hydroxypropyl)indoles

  2017cites this paper
• Iodine‐Catalyzed Azidation/Cyclization Cascade Approach to 3a‐Azidofuroindolines and ‐pyrroloindolines under Mild Conditions

  2017cites this paper
• Indole–Indole Ullmann Cross‐Coupling for CAr–N Bond Formation: Total Synthesis of (–)‐Aspergilazine A

  2017cites this paper
• Copper-Catalyzed Amination of Aryl and Alkenyl Electrophiles

  2017cites this paper
• Synthetic route to chiral indolines via Cu(OAc)2-catalyzed ring-opening/C(sp2)-H activation of activated aziridines.

  2017cites this paper
• Selenium-Iodine Cooperative Catalyst for Chlorocyclization of Tryptamine Derivatives.

  2017cites this paper
• Site-selective Cp*Rh(III)-catalyzed C–H amination of indolines with anthranils

  2017cites this paper
• The Diastereoselective Synthesis of Pyrroloindolines by Pd-Catalyzed Dearomative Cycloaddition of 1-Tosyl-2-vinylaziridine to 3-Nitroindoles

  2017cites this paper
• A Larock indolization approach to substituted tryptamines

  2017cites this paper
• Efficient oxidation of N-protected tryptophan and tryptophanyl-dipeptides by in situ generated dimethyldioxirane provides hexahydropyrroloindoline-containing synthons suitable for peptide synthesis and subsequent tryptathionylation

  2017cites this paper
• Total synthesis of naturally occurring (+)-psychotriasine and the related tetrahydro-β-carboline, dimeric tryptamines with NC connectivities

  2017cites this paper
• An asymmetric acetate-Mannich reaction of chiral isatin derived ketimines and its applications.

  2017cites this paper
• Lipase‐Catalyzed Kinetic Resolution of N‐Substituted 1‐(β‐Hydroxypropyl)indoles by Enantioselective Acetylation

  2017cites this paper
• Access to the Pyrroloindoline Core via [3 + 2] Annulation as well as the Application in the Synthetic Approach to (±)-Minfiensine.

  2016cites this paper
• Dearomatization through Halofunctionalization Reactions.

  2016cites this paper
• Synthesis of 2-oxindoles via 'transition-metal-free' intramolecular dehydrogenative coupling (IDC) of sp2 C–H and sp3 C–H bonds

  2016cites this paper
• Bioinspired Syntheses of the Pyridoacridine Marine Alkaloids Demethyldeoxyamphimedine, Deoxyamphimedine, and Amphimedine.

  2016cites this paper
• Marine AChE inhibitors isolated from Geodia barretti: natural compounds and their synthetic analogs.

  2016cites this paper
• A Mild and General Larock Indolization Protocol for the Preparation of Unnatural Tryptophans.

  2016cites this paper
• On the prevalence of bridged macrocyclic pyrroloindolines formed in regiodivergent alkylations of tryptophan

  2016cites this paper
• Asymmetric Mannich reaction: highly enantioselective synthesis of 3-amino-oxindoles via chiral squaramide based H-bond donor catalysis

  2016cites this paper
• Simple Synthesis of Multi‐Halogen Pyrazino[1,2‐a]indole‐1,8(2H,5aH)‐diones

  2016cites this paper
• A potent antibacterial indole alkaloid from Psychotria pilifera

  2016cites this paper
• Cutting-Edge and Time-Honored Strategies for Stereoselective Construction of C-N Bonds in Total Synthesis.

  2016cites this paper
• Lewis Acid Catalyzed Displacement of Trichloroacetimidates in the Synthesis of Functionalized Pyrroloindolines.

  2016cites this paper
• Synthetic approaches towards alkaloids bearing α-tertiary amines.

  2016cites this paper
• Reagent-switch controlled metal-free intermolecular geminal diamination and aminooxygenation of vinylarenes

  2016cites this paper
• Recent advances in the synthesis of benzimidazol(on)es via rearrangements of quinoxalin(on)es

  2016cites this paper
• N′-Acylation of (3,2′)-indole dimers

  2016cites this paper
• Stereodivergent and enantioselective total syntheses of isochaetominines A–C and four pairs of isochaetominine C enantiomers: a six-step approach

  2016cites this paper
• Stereoselective Anti‐Markovnikov Geminal Diamination and Dioxy­gena­tion of Vinylarenes Mediated by the Bromonium Ion

  2016cites this paper
• Rearrangements of Quinoxalin(on)es for the Synthesis of Benzimidazol(on)es

  2016cites this paper
• Enantioselective Synthesis of 3a-Amino-Pyrroloindolines by Copper-Catalyzed Direct Asymmetric Dearomative Amination of Tryptamines.

  2016cites this paper
• A Unified Approach to the Four Azaindoline Families by Inter-/Intramolecular Annulative Diamination of Vinylpyridines.

  2015cites this paper
• Synthesis and Biological Evaluation of Hexahydropyrrolo[2,3-b]Indole Derivatives as Fungicides against Phytopathogenic Fungi.

  2015cites this paper
• An organocatalytic Mannich/denitration reaction for the asymmetric synthesis of 3-ethylacetate-substitued 3-amino-2-oxindoles: formal synthesis of AG-041R.

  2015cites this paper
• Fluorescent kapakahines serve as non-toxic probes for live cell Golgi imaging.

  2015cites this paper
• Synthesis of naked amino-pyrroloindoline via direct aminocyclization of tryptamine.

  2015cites this paper
• Synthesis of Spirocyclic Pyrazolones by Oxidative C-N Bond Formation.

  2015cites this paper
• Total synthesis of the tetracyclic indole alkaloid ht-13-B.

  2015cites this paper
• Palladium-catalyzed intramolecular addition of C–N bond to alkynes: a novel approach to 3-diketoindoles

  2015cites this paper
• The Larock Reaction in the Synthesis of Heterocyclic Compounds

  2015cites this paper
• Total synthesis of the tetracyclic indole alkaloid ht-13-A

  2015cites this paper
• Advances in Dearomatization Strategies of Indoles

  2015cites this paper
• Enantioselective and diastereoselective azo-coupling/iminium-cyclizations: a unified strategy for the total syntheses of (–)-psychotriasine and (+)-pestalazine B

  2015cites this paper
• Iodohexahydropyridoindolones. Formation and reactivity

  2015cites this paper
• DMSO/Tf2O-mediated cross-coupling of tryptamine with substituted aniline to access C3a-N1'-linked pyrroloindoline alkaloids.

  2015cites this paper
• A Biomimetic Synthesis of Phaitanthrin E Involving a Fragmentation of sp(3) Carbon-Carbon Bond: Synthesis and Rearrangement of Phaitanthrin D to Phaitanthrin E.

  2015cites this paper
• Highly diastereoselective and regioselective copper-catalyzed nitrosoformate dearomatization reaction under aerobic-oxidation conditions.

  2014cites this paper
• Straightforward Access to Hexahydropyrrolo[2,3-b]indole Core by a Regioselective C3-Azo Coupling Reaction of Arenediazonium Compounds with Tryptamines.

  2014cites this paper
• Ruthenium-catalyzed synthesis of indoles from anilines and epoxides.

  2014cites this paper
• Natural product synthesis in the age of scalability.

  2014cites this paper
• Complexity generation by chemical synthesis: a five-step synthesis of (-)-chaetominine from L-tryptophan and its biosynthetic implications.

  2014cites this paper
• Synthetic approaches to 3-(2-nitroalkyl) indoles and their use to access tryptamines and related bioactive compounds.

  2014cites this paper
• Double annulative cascade of tryptophan-containing peptides triggered by selectfluor.

  2014cites this paper
• NIS-mediated regioselective amidation of indole with quinazolinone and pyrimidone

  2014cites this paper