Pharmacological characterisation of the presynaptic α-adrenoceptor in the rat vas deferens

No abstract is available for this paper.

• Publication year

  1977

• Venue

  European Journal of Pharmacology

• Publication date

  1977-03-21

• Fields of study

  Biology, Medicine, Chemistry

• Identifiers
  DOI 10.1016/0014-2999(77)90351-X
• External record

  Open on Semantic Scholar

• Source metadata

  Semantic Scholar

• No claims are published for this paper.

• No concepts are published for this paper.

• SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

  1997cited by this paper
• Effects of α-adrenoceptor agonists and antagonists on pre- and postsynaptically located α-adrenoceptors

  1976cited by this paper
• Inhibitory feedback modulation of adrenergic transmission.

  1975cited by this paper
• NORADRENALINE AND MOTOR TRANSMISSION IN THE VAS DEFERENS OF THE MOUSE

  1975cited by this paper
• Preferential blockade of presynaptic α-adrenoceptors by yohimbine

  1975cited by this paper
• Effects of lysergic acid diethylamide on autonomic post‐ganglionic transmission.

  1975cited by this paper
• REGIONAL VARIATION IN THE RESPONSE OF THE RAT VAS DEFERENS TO FIELD STIMULATION, TO NORADRENALINE AND TO TYRAMINE

  1974cited by this paper
• Negative feedback regulation of noradrenaline release by nerve stimulation in the perfused cat's spleen: differences in potency of phenoxybenzamine in blocking the pre‐ and post‐synaptic adrenergic receptors

  1974cited by this paper
• TRANSMISSION TO THE LONGITUDINAL MUSCLE OF THE GUINEA‐PIG VAS DEFERENS: THE EFFECT OF PRETREATMENT WITH GUANETHIDINE

  1974cited by this paper
• Presynaptic regulation of catecholamine release.

  1974cited by this paper
• An inhibition of post‐ganglionic motor transmission in the mammalian vas deferens by D‐lysergic acid diethylamide

  1973cited by this paper
• Inhibition of noradrenaline release by lysergic acid diethylamide

  1973cited by this paper
• Receptors for dopamine in some isolated vascular tissues of the dog.

  1972cited by this paper
• Evidence against adrenergic motor transmission in the guinea‐pig vas deferens

  1971cited by this paper
• Studies on neurotransmission mechanisms in the rat and guinea-pig vas deferens.

  1971cited by this paper
• The effects of adrenaline, noradrenaline and isoprenaline on inhibitory α‐ and β‐adrenoceptors in the longitudinal muscle of the guinea‐pig ileum

  1970cited by this paper
• The inhibitory action of noradrenaline and adrenaline on acetylcholine output by guinea‐pig ileum longitudinal muscle strip

  1969cited by this paper
• Competitive blockade of adrenergic α‐receptors and histamine receptors by thymoxamine

  1965cited by this paper
• The anticholinesterase activity of some antiadrenaline agents.

  1960cited by this paper

• Effects of clonidine in the isolated rat testicular capsule.

  2014cites this paper
• Binding sites of muscarinic and adrenergic receptors in gastrointestinal tissues of dairy cows suffering from left displacement of the abomasum.

  2010cites this paper
• Pharmacology of B-HT 920 in some isolated smooth muscles of the guinea-pig.

  2009cites this paper
• A New 2-Adrenoceptor Agonist with a1-Adrenoceptor Blocking Properties

  2009cites this paper
• EVIDENCE FOR oe-ADRENOCEPTOR TWO IN DISTINCTVASCULAR TYPES OF POSTSYNAPTIC SMOOTH MUSCLE in vivo

  2007cites this paper
• x-Adrenoceptor antagonism by apoyohimbine and some observations on the pharmacology of x-adrenoceptors in the rat anococcygeus and vas deferens

  2007cites this paper
• α1‐ and α2‐Adrenoreceptor Antagonist Profiles of 1‐ and 2‐[ω‐(4‐Arylpiperazin‐1‐yl)alkyl]‐1,2,3‐benzotriazoles

  2005cites this paper
• Antihypertensive effect of E-643, a new alpha-adrenergic blocking agent

  2004cites this paper
• Studies on YM-12617: A selective and potent antagonist of postsynaptic α1-adrenoceptors

  2004cites this paper
• Modifiers of gastrointestinal motility of cattle.

  2003cites this paper
• Searching for cyclazosin analogues as α1B-adrenoceptor antagonists

  2003cites this paper
• Structure--activity relationships among novel phenoxybenzamine-related beta-chloroethylamines.

  2002cites this paper
• Synthesis and α1-antagonist activity of derivatives of 4-chloro-5-{4-[2-(2-methoxyphenoxy)-ethyl]-1-piperazinyl}-3(2H)-pyridazinone

  2000cites this paper
• Comparative molecular field analysis of some pyridazinone-containing alpha1-antagonists.

  1999cites this paper
• AUTOINHIBITION, SYMPATHETIC COTRANSMISSION AND BIPHASIC CONTRACTILE RESPONSES TO TRAINS OF NERVE STIMULATION IN THE RODENT VAS DEFERENS

  1998cites this paper
• Synthesis and alpha-adrenoceptor blocking activity of the enantiomers of benzyl-(2-chloroethyl)-[2-(2-methoxyphenoxy)-1-methylethyl]amine hydrochloride.

  1997cites this paper
• Synthesis and α1-antagonist activity of new prazosin- and benextramine-related tetraamine disulfides

  1997cites this paper
• Enhanced α2A‐autoreceptor reserve for clonidine induced by reserpine and cholinomimetic agents in the rat vas deferens

  1997cites this paper
• Structure‐Activity Relationships of some 1,4‐Benzodioxane Aryl‐piperazine Derivatives as α‐Blocking Agents

  1997cites this paper
• Functional properties of agmatine in rat vas deferens.

  1996cites this paper
• Synthesis and alpha-adrenoreceptor blocking properties of phenoxybenzamine-related (2-chloroethyl)-(2,3-dihydrobenzo[1,4]dioxin- 2-ylmethyl)-(2-phenoxyethyl) amines.

  1995cites this paper
• Analysis of agonism at functional prejunctional alpha 2-adrenoceptors of rat vas deferens using operational and null approaches.

  1994cites this paper
• Effect of naringin and naringenin on contractions induced by noradrenaline in rat vas deferens--I. Evidence for postsynaptic alpha-2 adrenergic receptor.

  1993cites this paper
• Study of the mechanism of the relaxant action of (+)‐glaucine in rat vas deferens

  1993cites this paper
• Studyofthemechanism oftherelaxant action of(+)-glaucine inratvasdeferens

  1993cites this paper
• Acute and chronic effects of reserpine on biochemical and functional parameters of central and peripheral α2-adrenoceptors

  1993cites this paper
• Acute and chronic effects of cholinesterase inhibitors and pilocarpine on the density and sensitivity of central and peripheral α2-adrenoceptors

  1993cites this paper
• New pyridazinones: synthesis and correlation between structure and α-blocking activity

  1993cites this paper
• Modulation of α1‐adrenoceptors and functional consequences in the bisected rat vas deferens following chronic inhibition of neuronal noradrenaline uptake

  1993cites this paper
• Synthesis and Pharmacological Activity of Some New Pyridazinones

  1992cites this paper
• Stereoselectivity at alpha-adrenoreceptor subtypes: observations with the enantiomers of WB 4101 separated through their amides of N-tosyl-(S)-proline.

  1992cites this paper
• Inhibition of field stimulation-induced contractions of rat cauda epididymis by purinoceptor agonists but not by adrenoceptor agonists.

  1992cites this paper
• Release of contractile agents from rat vas deferens by clonidine.

  1991cites this paper
• Adrenoceptors of the human internal thoracic artery.

  1991cites this paper
• Clonidine-displacing substance (CDS) and its putative imidazoline receptor. New leads for further divergence of alpha 2-adrenergic receptor activity.

  1991cites this paper
• α2‐Adrenoceptor blocking profile of SK&F 104078: further evidence for receptor subtypes

  1991cites this paper
• Responses to noradrenaline in human subcutaneous resistance arteries are mediated by both α1‐ and α2‐adrenoceptors

  1990cites this paper
• Effects of St−587 on the α‐adrenoceptors in the Bisected Rat Vas Deferens

  1989cites this paper
• Calcium mobilization and phosphatidylinositol turnover in vas deferens smooth muscle of diabetic rats.

  1989cites this paper
• Inhibition of Ca‐spikes in rat preganglionic cervical sympathetic nerves by sympathomimetic amines

  1989cites this paper
• The pharmacology of α1- and α2-adrenoceptors: Evidence for and against a further subdivision

  1989cites this paper
• Fluoronorepinephrines: further pharmacological evaluation in vitro and in pithed rats.

  1987cites this paper
• Effects of methamphetamine on the twitch response in the rat isolated vas deferens.

  1987cites this paper
• The effects of some α-adrenoceptor antagonists on the responses of the canine saphenous vein to B-HT 933, UK-14304 and methoxamine

  1987cites this paper
• Electrophysiological evidence for an alpha 2-adrenergic inhibitory control of transmitter release in the rabbit mesenteric artery.

  1987cites this paper
• Pharmacological characterization of 5‐hydroxytryptamine‐induced hyperpolarization of the rat superior cervical ganglion

  1987cites this paper
• Two kinds of modification by 5-methoxy-N,N-dimethyltryptamine of contractile responses to electrical stimulation of isolated guinea-pig vas deferens.

  1987cites this paper
• Presynaptic α-autoreceptors

  1987cites this paper
• Resolution of the potent α1-adrenoreceptor antagonist 2-[[[2-(2,6-dimethoxyphenoxy)ethyl]amino]methyl]-1,4-benzoxathian (benoxathian)

  1987cites this paper
• 1 Pharmacology and Structure-Activity Relationships of α2-Adrenoceptor Antagonists

  1986cites this paper
• A study of the cardiovascular and respiratory pharmacology of amitraz

  1986influential citation
• Effects of putative α‐adrenoceptor antagonists and of other compounds on the loss of the righting reflex and on exophthalmia induced by xylazine in the rat

  1986cites this paper
• In vivo pharmacological activity of r 47 243 in rat: A comparison with putative α2‐adrenoceptor antagonists

  1986cites this paper
• Some pharmacological properties of Wy 27127 a more selective alpha2: alpha1-adrenoceptor antagonist than idazoxain in vitro

  1986cites this paper
• [Clinical and pharmacological studies on alpha-1 antagonists in smooth muscle of human urinary bladder base and prostatic urethra].

  1986cites this paper
• Probable pre- and postsynaptic modifications by 5-hydroxytryptamine of contractile responses to electrical stimulation of isolated guinea-pig vas deferens.

  1986cites this paper
• Compounds acting on alpha1‐ and alpha2‐ adrenoceptors: Agonists and antagonists

  1986cites this paper
• SELECTIVITIES OF SOME AGONISTS ACTING AT α1‐ AND α2‐ADRENORECEPTORS IN THE RAT VAS DEFERENS

  1986cites this paper
• The effect of age on the sensitivity of pre- and postsynaptic alpha-adrenoceptors to agonists and antagonists in the rat

  1986cites this paper
• L-654,284 a new potent and selective α2-adrenoceptor antagonist

  1986cites this paper
• Distribution of Presynaptic Receptors Modulating Acetylcholine Release

  1986cites this paper
• Activation and desensitization of presynaptic α2‐adrenoceptors after inhibition of neuronal uptake by antidepressant drugs in the rat vas deferens

  1986cites this paper
• Differential blocking actions of idazoxan against the inhibitory effects of 6‐fluoronoradrenaline and clonidine in the rat vas deferens

  1985cites this paper
• Mechanism of action of B-HT 933 (azepexole) in rat vas deferens and guinea-pig ileum.

  1985cites this paper
• Presynaptic regulation by ACh of the NE mediated responses in the rat vas deferens.

  1985cites this paper
• Opiatentzug und α2-Stimulation Prinzipielle Möglichkeiten (Clonidin und Analoge)

  1985cites this paper
• A difference in the affinity of some selective α2-adrenoceptor antagonists when compared on isolated vasa deferentia of rat and rabbit

  1985cites this paper
• Evaluation of the α1- and α2-adrenoceptor effects of detomidine, a novel veterinary sedative analgesic

  1985cites this paper
• Effect of some smooth muscle stimulants and trypsin on the contraction of vas deferens of aging rats.

  1985cites this paper
• Alpha-adrenolytic properties of apogalanthamine and azapetine analogs.

  1985cites this paper
• Differences between the prejunctional effects of phenylephrine and clonidine in guinea‐pig isolated atria

  1984cites this paper
• The mechanism of action of dopamine to inhibit field stimulation-induced contractions of guinea pig stomach strips

  1984cites this paper
• Alpha2-adrenoceptor antagonism and other pharmacological antagonist properties of some substituted benzoquinolizines and yohimbine in vitro

  1984cites this paper
• α‐Adrenoceptor antagonism by apoyohimbine and some observations on the pharmacology of α‐adrenoceptors in the rat anococcygeus and vas deferens

  1984cites this paper
• The action and interaction of β‐phenethylamines and imidazolines on prejunctional α2‐adrenoceptors of guinea‐pig ileum in the presence of the non‐competitive antagonist benextramine

  1984cites this paper
• Interaction between 2-chloroadenosine and α-adrenoceptors in rat vas deferens

  1984cites this paper
• Presynaptic agonist effect of phentolamine in the rabbit vas deferens and rat cerebral cortex

  1984cites this paper
• Non‐specific, time‐dependent desensitization of the vas deferens and anococcygeus preparations of the rat to α1‐adrenoceptor antagonists and atropine

  1984cites this paper
• Separation of adrenergic and non‐adrenergic contractions to field stimulation in the rat vas deferens

  1983cites this paper
• Pharmacological characterization of postjunctional alpha-adrenoceptors in isolated feline cerebral and peripheral arteries.

  1983cites this paper
• Microelectrode recording of the effects of agonists and antagonists on α‐adrenoceptors on rat somatic nerve terminals

  1983influential citation
• Cardiovascular α2-receptors

  1983cites this paper
• The use of neurally released agonist in the measurement of antagonism at α‐adrenoceptors

  1983cites this paper
• Characterization of postsynaptic α‐adrenoceptors in rat aortic strips and portal veins

  1983cites this paper
• Effect of thymoxamine on the human pupil.

  1983cites this paper
• A STUDY OF STIMULATION‐EVOKED ACTIVATION OF α2‐ADRENOCEPTORS IN THE RAT ISOLATED VAS DEFERENS

  1983cites this paper
• Feedback inhibition of responses of rat vas deferens to twin pulse stimulation.

  1983cites this paper
• Benzamide action at α2-adrenoceptors modifies catecholamine-induced contraction and relaxation of circular smooth muscle from guinea-pig stomach

  1982cites this paper
• Pre‐ and postsynaptic effects of sulpiride in the rat isolated vas deferens

  1982cites this paper
• Acebutolol: A Review of its Pharmacology, Pharmacokinetics, Clinical Uses, and Adverse Effects

  1982cites this paper
• Functional postsynaptic α2- but not α1-adrenoceptors in dog saphenous vein exposed to phenoxybenzamine

  1982cites this paper
• Interactions between the autonomic nervous system and the cardiovascular effects of ouabain in guinea-pigs.

  1982cites this paper
• High and low (Gpp(NH)p-sensitive) affinity sites for beta 2-adrenergic blockers as antagonists of isoproterenol in the field-stimulated rat vas deferens.

  1982cites this paper
• Catecholamine‐induced relaxation and contraction of the lower oesophageal and pyloric sphincters of guinea‐pig stomach: modification by domperidone

  1982cites this paper
• Catecholamines act at α2‐adrenoceptors to cause contraction of circular smooth muscle of guinea‐pig stomach

  1982cites this paper
• Effects of prazosin and piperoxan on central cardiovascular actions of St 91 in cats.

  1982cites this paper
• Evidence for more than one type of post-junctional α-Adrenoceptor

  1982cites this paper
• Modulation of central noradrenaline release by postsynaptic receptors

  1982cites this paper
• Antihypertensive and adrenoceptor blocking properties of new sulfonamide-substituted phenylethylamines.

  1982cites this paper
• Development of clonidine-tolerance in the rat vas deferens: cross tolerance to other presynaptic inhibitory agents.

  1982cites this paper